SCHEMBL4013386

SCHEMBL4013386

COc1cccc2c(-c3cc(OS(=O)(=O)C(F)(F)F)ccc3Cl)ccnc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.39
NR1H2 P55055 7/20 0.39
NR1H3 Q13133 7/20 0.39
HTR1A P08908 2/20 0.39
ADRA1D P25100 2/20 0.39
ADRA1A P35348 2/20 0.39
ADRA1B P35368 2/20 0.39
RXRA P19793 1/20 0.38
PDE4A P27815 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
CCNT1 O60563 1/20 0.36
CDK9 P50750 1/20 0.36
ENPP3 O14638 1/20 0.36
ENPP1 P22413 1/20 0.36
SLC40A1 Q9NP59 1/20 0.36
MAPK14 Q16539 1/20 0.36
KMT2A Q03164 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4018578 0.88 PTGDR2 (0.41) PTGDR2NR1H2NR1H3HTR1AADRA1D
SCHEMBL4012080 0.88 NR1H2 (0.47) PTGDR2NR1H2NR1H3HTR1ARXRA
SCHEMBL4012347 0.85 NR1H3 (0.45) PTGDR2NR1H2NR1H3HTR1ARXRA
SCHEMBL4013308 0.84 HTR1A (0.47) PTGDR2NR1H2NR1H3HTR1AADRA1D
SCHEMBL4010967 0.84 NR1H2 (0.53) PTGDR2NR1H2NR1H3HTR1AADRA1D
SCHEMBL4017522 0.80 NR1H2 (0.45) PTGDR2NR1H2NR1H3HTR1ARXRA
SCHEMBL4011491 0.80 NR1H2 (0.64) NR1H2NR1H3RXRACDK9
SCHEMBL4010720 0.78 NR1H2 (0.52) PTGDR2NR1H2NR1H3HTR1AADRA1D
SCHEMBL4013490 0.78 NR1H2 (0.52) NR1H2NR1H3RXRAMAPK14
SCHEMBL4012811 0.77 NR1H2 (0.53) PTGDR2NR1H2NR1H3HTR1AADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed