SCHEMBL4016970

SCHEMBL4016970

CS(=O)(=O)c1cccc2c(-c3cc(OS(=O)(=O)C(F)(F)F)ccc3F)ccnc12

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR1H3 Q13133 10/20 0.50
NR1H2 P55055 9/20 0.50
PTGDR2 Q9Y5Y4 1/20 0.43
RXRA P19793 1/20 0.42
PDE4A P27815 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
CHRM1 P11229 4/20 0.35
DRD2 P14416 4/20 0.35
DRD4 P21917 4/20 0.35
DRD3 P35462 4/20 0.35
GLO1 Q04760 1/20 0.35
HTR1A P08908 1/20 0.34
HTR1D P28221 1/20 0.34
HTR1B P28222 1/20 0.34
CCNT1 O60563 1/20 0.34
CDK9 P50750 1/20 0.34
GCK P35557 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4012347 0.88 NR1H3 (0.45) NR1H3NR1H2PTGDR2RXRAPDE4A
SCHEMBL4010255 0.87 NR1H2 (0.48) NR1H3NR1H2PTGDR2RXRAPDE4A
SCHEMBL4018578 0.85 PTGDR2 (0.41) NR1H3NR1H2PTGDR2RXRAPDE4A
SCHEMBL4017522 0.85 NR1H2 (0.45) NR1H3NR1H2PTGDR2RXRAPDE4A
SCHEMBL4011973 0.82 NR1H2 (0.58) NR1H3NR1H2PTGDR2RXRA
SCHEMBL4299566 0.80 NR1H2 (0.50) NR1H3NR1H2PTGDR2RXRAGLO1
SCHEMBL4010387 0.80 NR1H2 (0.48) NR1H3NR1H2PTGDR2RXRAGCK
SCHEMBL4012970 0.79 NR1H2 (0.52) NR1H3NR1H2PTGDR2RXRAGCK
SCHEMBL4017675 0.79 NR1H2 (0.50) NR1H3NR1H2PTGDR2RXRA
SCHEMBL4011406 0.79 CYP4F2 (0.44) NR1H3NR1H2PTGDR2RXRAPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed