SCHEMBL4012780

SCHEMBL4012780

Cc1cc(-c2cc(O)ccc2F)c2cccc(C(F)(F)F)c2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD38 P28907 4/20 0.41
CYP3A4 P08684 2/20 0.41
KCNH2 Q12809 1/20 0.41
ESR1 P03372 4/20 0.41
GAA P10253 2/20 0.40
MAPT P10636 1/20 0.40
ACVR1 Q04771 1/20 0.38
NR1H2 P55055 2/20 0.37
NR1H3 Q13133 2/20 0.37
HSD17B1 P14061 1/20 0.37
HSD17B2 P37059 1/20 0.37
ALDH1A1 P00352 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
SRC P12931 1/20 0.36
SYK P43405 1/20 0.36
ESR2 Q92731 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
TP53 P04637 1/20 0.35
MGAM O43451 1/20 0.34
SI P14410 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4012143 0.86 ESR1 (0.40) CD38CYP3A4ESR1GAAMAPT
SCHEMBL4019153 0.83 NR4A2 (0.50) CD38CYP3A4GAAMAPTL3MBTL1
SCHEMBL4015511 0.82 ENPP1 (0.40) CD38CYP3A4KCNH2ESR1GAA
SCHEMBL4014169 0.82 PIK3CD (0.46) CD38CYP3A4KCNH2ESR1GAA
SCHEMBL4010284 0.81 NR1H2 (0.53) ESR1NR1H2NR1H3L3MBTL1
SCHEMBL4014835 0.78 NR1H2 (0.39) CD38CYP3A4KCNH2ESR1ACVR1
SCHEMBL4012475 0.76 NR1H2 (0.58) NR1H2NR1H3
SCHEMBL9494183 0.76 CD38 (0.44) CD38CYP3A4KCNH2ESR1GAA
SCHEMBL2446200 0.74 ESR1 (0.41) ESR1NR1H2NR1H3HSD17B1HSD17B2
SCHEMBL4012268 0.74 NR1H2 (0.58) NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed