SCHEMBL4013099

SCHEMBL4013099

O=C1NCCN1c1cccc(CBr)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.45
CYP2C19 P33261 2/20 0.45
HTR1A P08908 2/20 0.45
HTR1D P28221 2/20 0.45
HTR1B P28222 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
DRD2 P14416 1/20 0.45
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45
HTR7 P34969 1/20 0.45
DRD3 P35462 1/20 0.45
HTR2B P41595 1/20 0.45
KCNH2 Q12809 1/20 0.45
POLB P06746 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
MAPT P10636 1/20 0.43
ALOX5 P09917 5/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4018203 0.93 ALOX5 (0.47) CYP2C9CYP2C19HTR1AHTR1DHTR1B
SCHEMBL27765059 0.88 CYP2C9 (0.48) CYP2C9CYP2C19HTR1AHTR1DHTR1B
SCHEMBL27765009 0.84 ALOX5 (0.52) CYP2C9CYP2C19HTR1AHTR1DHTR1B
SCHEMBL13853418 0.84 CYP2C9 (0.45) CYP2C9CYP2C19HTR1AHTR1DHTR1B
Hydrochloric Acid SCHEMBL3950851 0.83 CYP2C9 (0.44) CYP2C9CYP2C19HTR1AHTR1DHTR1B
SCHEMBL7011655 0.82 CYP2C9 (0.43) CYP2C9CYP2C19HTR1AHTR1DHTR1B
SCHEMBL2885321 0.82 HTR1A (0.48) CYP2C9CYP2C19HTR1AHTR1DHTR1B
SCHEMBL2878333 0.81 ITGB3 (0.48) CYP2C9CYP2C19HTR1AHTR1DHTR1B
SCHEMBL31731890 0.79 CRBN (0.64) ALOX5DDB1CRBNALDH1A1
SCHEMBL1787047 0.79 ALDH1A1 (0.51) MEN1KMT2AALOX5DDB1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed