SCHEMBL4013470

SCHEMBL4013470

Cc1cc(NC(=O)NCCN2CCC(CNS(=O)(=O)c3ccccc3)CC2)cc(C)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.54
L3MBTL1 Q9Y468 1/20 0.48
PKM P14618 1/20 0.47
RAB9A P51151 1/20 0.46
CCR3 P51677 3/20 0.46
GBA1 P04062 1/20 0.46
OPRM1 P35372 1/20 0.45
OPRK1 P41145 1/20 0.45
HDAC3 O15379 2/20 0.45
HDAC4 P56524 2/20 0.45
HDAC1 Q13547 2/20 0.45
HDAC7 Q8WUI4 2/20 0.45
HDAC2 Q92769 2/20 0.45
HDAC10 Q969S8 2/20 0.45
HDAC11 Q96DB2 2/20 0.45
HDAC8 Q9BY41 2/20 0.45
HDAC6 Q9UBN7 2/20 0.45
HDAC9 Q9UKV0 2/20 0.45
HDAC5 Q9UQL6 2/20 0.45
MEN1 O00255 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4017971 0.92 RAB9A (0.46) ALDH1A1RAB9ACCR3OPRM1OPRK1
SCHEMBL3565136 0.90 ALDH1A1 (0.51) ALDH1A1MEN1POLBKMT2ANAMPT
SCHEMBL4016844 0.83 MAPT (0.45) PKMCCR3KMT2AMAPT
SCHEMBL3557299 0.82 CCR3 (0.67) RAB9ACCR3MEN1POLBKMT2A
SCHEMBL3565549 0.81 HTR2A (0.49) L3MBTL1MEN1POLBKMT2ANAMPT
SCHEMBL3565154 0.81 UTS2R (0.46) ALDH1A1RAB9ACCR3MEN1POLB
SCHEMBL3564763 0.81 NAMPT (0.47) RAB9ACCR3MEN1POLBKMT2A
SCHEMBL3557010 0.80 CARM1 (0.52) ALDH1A1RAB9AMEN1POLBKMT2A
SCHEMBL3559283 0.77 RAB9A (0.44) RAB9ACCR3MEN1POLBKMT2A
SCHEMBL301872 0.77 NAMPT (0.47) PKMCCR3MEN1POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1670470-B1 PYRIDINE DERIVATIVES AND USE THEREOF AS UROTENSIN II ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2009-04-08 EP disclosed