SCHEMBL4013567

SCHEMBL4013567

COc1cccc2c(-c3cccc(O)c3)ccnc12

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.57
FYN P06241 5/20 0.49
HTR1A P08908 2/20 0.49
ADRA1D P25100 2/20 0.49
ADRA1A P35348 2/20 0.49
ADRA1B P35368 2/20 0.49
PTGDR2 Q9Y5Y4 1/20 0.44
CDC7 O00311 1/20 0.44
BMPR1A P36894 1/20 0.43
TGFBR1 P36897 1/20 0.43
ACVRL1 P37023 1/20 0.43
ACVR1 Q04771 1/20 0.43
HSD17B1 P14061 1/20 0.43
HSD17B2 P37059 1/20 0.43
DYRK1A Q13627 2/20 0.41
RAF1 P04049 2/20 0.41
TOP2A P11388 1/20 0.41
PDE10A Q9Y233 1/20 0.40
ACACA Q13085 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4011409 0.81 PIK3CD (0.61) PIK3CDHTR1AADRA1DADRA1AADRA1B
SCHEMBL4016936 0.80 HTR1A (0.46) PIK3CDHTR1AADRA1DADRA1AADRA1B
SCHEMBL4013847 0.80 MAPK14 (0.46) PIK3CDFYNHTR1AADRA1DADRA1A
SCHEMBL30275434 0.80 HTR1A (0.54) HTR1AADRA1DADRA1AADRA1BPTGDR2
SCHEMBL25289806 0.80 HTR1A (0.54) HTR1AADRA1DADRA1AADRA1BPTGDR2
SCHEMBL4013369 0.78 PIK3CD (0.65) PIK3CDFYNPTGDR2CDC7HSD17B1
SCHEMBL4016535 0.78 PIK3CD (0.61) PIK3CDHTR1APTGDR2CDC7HSD17B1
SCHEMBL6558762 0.78 PIK3CD (0.60) PIK3CDCDC7ACVR1HSD17B1HSD17B2
SCHEMBL1125582 0.78 NR1H2 (0.62) PIK3CDPTGDR2CDC7HSD17B1HSD17B2
SCHEMBL4013993 0.77 NR1H2 (0.68) HTR1AADRA1DADRA1AADRA1BACVR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101541751-A Quinoline compounds WYETH CORP (US) 2009-09-23 CN disclosed
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed