SCHEMBL4016936

SCHEMBL4016936

COc1cccc2c(-c3cc(O)ccc3Cl)ccnc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.46
ADRA1D P25100 2/20 0.46
ADRA1A P35348 2/20 0.46
ADRA1B P35368 2/20 0.46
PTGDR2 Q9Y5Y4 1/20 0.42
PDE4D Q08499 4/20 0.41
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
RET P07949 1/20 0.40
KIF5B P33176 1/20 0.40
KDR P35968 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
G6PD P11413 1/20 0.39
ATP4A P20648 2/20 0.39
ATP4B P51164 2/20 0.39
NQO2 P16083 1/20 0.39
MAPK14 Q16539 1/20 0.39
KDM4E B2RXH2 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4013308 0.86 HTR1A (0.47) HTR1AADRA1DADRA1AADRA1BPTGDR2
SCHEMBL4013847 0.85 MAPK14 (0.46) HTR1AADRA1DADRA1AADRA1BPTGDR2
SCHEMBL4011946 0.84 NR4A2 (0.49) HTR1APTGDR2PDE4DMAPK14KDM4E
SCHEMBL3509876 0.82 RET (0.43) HTR1AADRA1DADRA1AADRA1BRET
SCHEMBL4013567 0.80 PIK3CD (0.57) HTR1AADRA1DADRA1AADRA1BPTGDR2
SCHEMBL4009254 0.80 NR1H2 (0.47) HTR1APTGDR2PDE4DMAPK14KDM4E
SCHEMBL4012181 0.78 PTGDR2 (0.45) HTR1APTGDR2PDE4DNPC1RAB9A
SCHEMBL4020656 0.77 PTGDR2 (0.41) HTR1APTGDR2PDE4DMAPK14KDM4E
SCHEMBL4013386 0.76 PTGDR2 (0.39) HTR1AADRA1DADRA1AADRA1BPTGDR2
SCHEMBL4011501 0.76 NR1H2 (0.55) HTR1AADRA1DADRA1AADRA1BKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed