SCHEMBL4013817

SCHEMBL4013817

Cc1cc(-c2cccc(O)c2)c2cccc(Cl)c2n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 4/20 0.54
PIK3CD O00329 1/20 0.48
CRHR1 P34998 2/20 0.42
DHODH Q02127 1/20 0.41
HSD17B2 P37059 4/20 0.41
HSD17B1 P14061 3/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
MAPT P10636 2/20 0.40
GAA P10253 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PARP1 P09874 1/20 0.39
PRKAB2 O43741 1/20 0.39
PRKAG1 P54619 1/20 0.39
PRKAA2 P54646 1/20 0.39
PRKAA1 Q13131 1/20 0.39
PRKAG3 Q9UGI9 1/20 0.39
PRKAG2 Q9UGJ0 1/20 0.39
PRKAB1 Q9Y478 1/20 0.39
MGAM O43451 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28046875 0.85 NR4A2 (0.59) NR4A2CRHR1DHODHMAPTL3MBTL1
SCHEMBL4017818 0.83 NR4A2 (0.54) NR4A2CRHR1MAPTGAAL3MBTL1
SCHEMBL4014169 0.81 PIK3CD (0.46) PIK3CDHSD17B2HSD17B1CYP3A4MAPT
SCHEMBL4019153 0.80 NR4A2 (0.50) NR4A2CRHR1CYP3A4MAPTGAA
SCHEMBL1026984 0.77 NR4A2 (0.65) NR4A2CRHR1DHODHCYP3A4MAPT
SCHEMBL4016535 0.77 PIK3CD (0.61) NR4A2PIK3CDHSD17B2HSD17B1CYP3A4
Phenol SCHEMBL28074113 0.75 KDM4E (0.45) PIK3CDCRHR1HSD17B2HSD17B1CYP2C9
SCHEMBL3063558 0.74 NR4A2 (0.71) NR4A2CRHR1DHODHCYP3A4MAPT
SCHEMBL28176160 0.74 HSD17B1 (0.47) CRHR1DHODHHSD17B2HSD17B1CYP2C9
SCHEMBL4018305 0.73 NR1H2 (0.45) NR4A2CRHR1DHODHPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed