SCHEMBL4016329

SCHEMBL4016329

Cc1ccc(OC(=O)NC(C)(C)C)cc1N

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.42
MAPT P10636 2/20 0.42
ACHE P22303 5/20 0.41
BCHE P06276 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.36
ALDH1A1 P00352 3/20 0.36
CASP1 P29466 1/20 0.36
LMNA P02545 1/20 0.35
NPC1 O15118 2/20 0.35
KDM4E B2RXH2 1/20 0.35
RAB9A P51151 1/20 0.35
CYP3A4 P08684 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NR1H4 Q96RI1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28032033 0.88 ACHE (0.44) TDP1MAPTACHEBCHESMN1; SMN2
SCHEMBL29286667 0.83 ACHE (0.40) MAPTACHEBCHESMN1; SMN2LMNA
SCHEMBL27760985 0.81 RAB9A (0.41) MAPTACHEBCHESMN1; SMN2ALDH1A1
SCHEMBL27470803 0.80 ACHE (0.43) MAPTACHEBCHEALDH1A1CASP1
SCHEMBL29000949 0.79 ACHE (0.42) TDP1MAPTACHEBCHESMN1; SMN2
SCHEMBL28043917 0.79 ALDH1A1 (0.51) TDP1ACHEBCHEALDH1A1LMNA
SCHEMBL5510119 0.79 ELANE (0.55) TDP1MAPT
SCHEMBL3813706 0.78 MAPT (0.51) TDP1MAPTACHEBCHESMN1; SMN2
SCHEMBL4573467 0.78 ACHE (0.41) ACHEBCHENR1H4
SCHEMBL2314345 0.78 TSHR (0.48) TDP1MAPTACHEBCHESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009089042-A1 PYRAZOLE PYRAZINE AMINE COMPOUNDS AS KINASE INHIBITORS, COMPOSITIONS THEREOF AND METHODS OF TREATMENT THEREWITH SIGNAL PHARMACEUTICALS, LLC (US) 2009-07-16 WO disclosed
CN-101421262-A Compounds and compositions as protein kinase inhibitors IRM LLC (VG) 2009-04-29 CN disclosed