SCHEMBL4016601

SCHEMBL4016601

N#Cc1cccc2c(-c3cccc(O)c3)ccnc12

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.57
LRRK2 Q5S007 5/20 0.56
CDC7 O00311 1/20 0.44
PTGDR2 Q9Y5Y4 1/20 0.43
AR P10275 1/20 0.42
GSK3B P49841 1/20 0.41
DYRK1A Q13627 1/20 0.41
NUDT1 P36639 1/20 0.40
TOP2A P11388 1/20 0.39
HSD17B1 P14061 1/20 0.38
HSD17B2 P37059 1/20 0.38
IKBKB O14920 1/20 0.38
CHUK O15111 1/20 0.38
ADORA2A P29274 1/20 0.37
ADORA2B P29275 1/20 0.37
ADORA1 P30542 1/20 0.37
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37
CYP19A1 P11511 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4020656 0.80 PTGDR2 (0.41) PIK3CDLRRK2PTGDR2ARGSK3B
SCHEMBL4011409 0.78 PIK3CD (0.61) PIK3CDLRRK2CDC7PTGDR2DYRK1A
SCHEMBL4016535 0.78 PIK3CD (0.61) PIK3CDLRRK2CDC7PTGDR2NUDT1
SCHEMBL4013369 0.78 PIK3CD (0.65) PIK3CDLRRK2CDC7PTGDR2TOP2A
SCHEMBL6558762 0.78 PIK3CD (0.60) PIK3CDLRRK2CDC7DYRK1ATOP2A
SCHEMBL4012471 0.76 KDM4E (0.42) LRRK2PTGDR2ARGSK3BDYRK1A
SCHEMBL4013567 0.75 PIK3CD (0.57) PIK3CDCDC7PTGDR2DYRK1ATOP2A
SCHEMBL1125582 0.75 NR1H2 (0.62) PIK3CDCDC7PTGDR2ARGSK3B
SCHEMBL1028218 0.74 ESR2 (0.65) LRRK2ARHSD17B1HSD17B2ADORA2A
SCHEMBL23832886 0.73 HTT (0.46) LRRK2PTGDR2ARGSK3BDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101541751-A Quinoline compounds WYETH CORP (US) 2009-09-23 CN disclosed
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed