SCHEMBL4012471

SCHEMBL4012471

N#Cc1cccc2c(O)ccnc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.42
LMNA P02545 2/20 0.42
MAPT P10636 2/20 0.42
TP53 P04637 1/20 0.42
TSHR P16473 1/20 0.42
ALOX12 P18054 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.40
KDM4A O75164 1/20 0.40
RAB9A P51151 1/20 0.40
EGLN1 Q9GZT9 1/20 0.40
HIF1AN Q9NWT6 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.40
AR P10275 6/20 0.39
HTT P42858 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
LRRK2 Q5S007 1/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
CA1 P00915 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4608765 0.86 LMNA (0.49) KDM4ELMNAMAPTALOX12L3MBTL1
SCHEMBL23832886 0.83 HTT (0.46) KDM4EMAPTPTGDR2ARHTT
SCHEMBL317372 0.79 KDM4E (0.49) KDM4ELMNAMAPTTP53ALOX12
SCHEMBL3156281 0.79 PSMD14 (0.56) TSHRL3MBTL1PTGDR2ARHTT
SCHEMBL667933 0.79 HTT (0.42) KDM4EMAPTTP53PTGDR2AR
SCHEMBL10008410 0.79 NR4A2 (0.56) TSHRPTGDR2ARHTTLRRK2
SCHEMBL28906978 0.79 KDM4E (0.54) KDM4ELMNAMAPTTP53TSHR
SCHEMBL7641703 0.77 KDM4E (0.62) KDM4EL3MBTL1KDM4ARAB9AEGLN1
SCHEMBL30668494 0.77 KDM4E (0.66) KDM4ELMNAMAPTTP53TSHR
SCHEMBL1333120 0.77 KDM4E (0.66) KDM4ELMNAMAPTTP53TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119899214-A Iridium-containing Lewis base catalyst and preparation method and application thereof 山东汇盟生物科技股份有限公司 2025-04-29 CN claimed
EP-4055014-B1 PYRROLIDINE AND PIPERIDINE COMPOUNDS YUHAN CORP (KR) 2025-04-30 EP disclosed
CN-119899214-A Iridium-containing Lewis base catalyst and preparation method and application thereof 山东汇盟生物科技股份有限公司 2025-04-29 CN disclosed
CN-119798315-A Preparation method of L-smart glufosinate 山东汇盟生物科技股份有限公司 2025-04-11 CN disclosed
CN-114867719-B Pyrrolidine and piperidine compounds 柳韩洋行 2024-06-25 CN disclosed
US-11655235-B2 Pyrrolidine and piperidine compounds YUHAN CORPORATION (KR) 2023-05-23 US disclosed
EP-4055014-A1 PYRROLIDINE AND PIPERIDINE COMPOUNDS Yuhan Corporation (KR) 2022-09-14 EP disclosed
CN-114867719-A Pyrrolidine and piperidine compounds 柳韩洋行 2022-08-05 CN disclosed
US-20210147386-A1 PYRROLIDINE AND PIPERIDINE COMPOUNDS YUHAN CORPORATION (KR) 2021-05-20 US disclosed
CN-101541751-A Quinoline compounds WYETH CORP (US) 2009-09-23 CN disclosed
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11655235-B2 Pyrrolidine and piperidine compounds FAP, APC, VHL KDM4E 1644/4885LMNA 1955/4885MAPT 1909/4885
US-20210147386-A1 PYRROLIDINE AND PIPERIDINE COMPOUNDS FAP, APC, VHL KDM4E 1644/4885LMNA 1955/4885MAPT 1909/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.