SCHEMBL4016946

SCHEMBL4016946

COc1ccc(F)c(-c2ccnc3c(OC)cccc23)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.47
ADRA1D P25100 2/20 0.47
ADRA1A P35348 2/20 0.47
ADRA1B P35368 2/20 0.47
MAPK14 Q16539 3/20 0.47
PTGDR2 Q9Y5Y4 1/20 0.43
RAB9A P51151 2/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
THRB P10828 1/20 0.41
BLM P54132 1/20 0.41
CASP6 P55212 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TRPA1 O75762 3/20 0.41
TGFBR1 P36897 2/20 0.40
ATR Q13535 1/20 0.39
ATRIP Q8WXE1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4013847 0.86 MAPK14 (0.46) HTR1AADRA1DADRA1AADRA1BMAPK14
SCHEMBL4018578 0.85 PTGDR2 (0.41) HTR1AADRA1DADRA1AADRA1BMAPK14
SCHEMBL4012417 0.85 NR1H2 (0.51) MAPK14PTGDR2ATRATRIPCYP1A2
SCHEMBL4013308 0.84 HTR1A (0.47) HTR1AADRA1DADRA1AADRA1BMAPK14
SCHEMBL4010852 0.83 NR1H2 (0.56) MAPK14
SCHEMBL4010255 0.82 NR1H2 (0.48) MAPK14PTGDR2POLBMAPTKMT2A
SCHEMBL4017304 0.81 NR1H2 (0.46) HTR1AADRA1DADRA1AADRA1BMAPK14
SCHEMBL4011231 0.80 NR1H2 (0.47) MAPK14PTGDR2
SCHEMBL4011122 0.80 NR1H2 (0.58) HTR1AADRA1DADRA1AADRA1BMAPK14
SCHEMBL30365370 0.80 MAPK14 (0.55) HTR1AADRA1DADRA1AADRA1BMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed