SCHEMBL4013308

SCHEMBL4013308

COc1ccc(Cl)c(-c2ccnc3c(OC)cccc23)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.47
ADRA1D P25100 2/20 0.47
ADRA1A P35348 2/20 0.47
ADRA1B P35368 2/20 0.47
CCNT1 O60563 2/20 0.44
CDK9 P50750 2/20 0.44
ALDH1A1 P00352 2/20 0.41
POLB P06746 2/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
THRB P10828 1/20 0.41
RAB9A P51151 1/20 0.41
BLM P54132 1/20 0.41
CASP6 P55212 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
ENPP3 O14638 1/20 0.40
ENPP1 P22413 1/20 0.40
G6PD P11413 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4017565 0.89 NR1H2 (0.47) CCNT1CDK9ALDH1A1MEN1KMT2A
SCHEMBL4016936 0.86 HTR1A (0.46) HTR1AADRA1DADRA1AADRA1BALDH1A1
SCHEMBL4013386 0.84 PTGDR2 (0.39) HTR1AADRA1DADRA1AADRA1BCCNT1
SCHEMBL4016946 0.84 HTR1A (0.47) HTR1AADRA1DADRA1AADRA1BALDH1A1
SCHEMBL4013857 0.84 NR1H2 (0.47) CCNT1CDK9MAPTRAB9APTGDR2
SCHEMBL4011959 0.83 LRRK2 (0.42) CCNT1CDK9ALDH1A1MEN1MAPT
SCHEMBL4011491 0.83 NR1H2 (0.64) CDK9CLK4NR1H2NR1H3
SCHEMBL4011482 0.82 NR1H2 (0.47) CCNT1CDK9ALDH1A1POLBMEN1
SCHEMBL4010720 0.81 NR1H2 (0.52) HTR1AADRA1DADRA1AADRA1BPOLB
SCHEMBL4012811 0.80 NR1H2 (0.53) HTR1AADRA1DADRA1AADRA1BCCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed