SCHEMBL4017325

SCHEMBL4017325

O=C1OCCN1c1cccc(CO)c1.OCc1cccc(Br)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.42
HTR1A P08908 2/20 0.42
HTR1D P28221 2/20 0.42
HTR1B P28222 2/20 0.42
DRD2 P14416 1/20 0.42
HTR2A P28223 1/20 0.42
HTR7 P34969 1/20 0.42
DRD3 P35462 1/20 0.42
HTR2B P41595 1/20 0.42
HTR6 P50406 1/20 0.42
KCNH2 Q12809 1/20 0.42
HSD11B1 P28845 1/20 0.41
KDM1A O60341 2/20 0.40
MAOA P21397 2/20 0.40
MAOB P27338 2/20 0.40
KDM1B Q8NB78 2/20 0.40
RCOR1 Q9UKL0 2/20 0.40
FAAH O00519 2/20 0.38
NAAA Q02083 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4017984 0.88 ALOX5 (0.43) ALOX5HTR1AHTR1DHTR1BDRD2
SCHEMBL4004501 0.85 HSD11B1 (0.52) ALOX5HTR1AHTR1DHTR1BDRD2
SCHEMBL2882743 0.81 HTR1A (0.49) HTR1AHTR1DHTR1BDRD2HTR2A
SCHEMBL4018668 0.81 HTR1A (0.46) HTR1AHTR1DHTR1BDRD2HTR2A
SCHEMBL8413923 0.79 HTR1A (0.49) HTR1AHTR1DHTR1BDRD2HTR2A
SCHEMBL7904237 0.78 MGLL (0.50) ALOX5HTR1AHTR1DHTR1BDRD2
SCHEMBL13853420 0.78 HTR1A (0.46) HTR1AHTR1DHTR1BDRD2HTR2A
SCHEMBL2883416 0.77 HTR1A (0.45) HTR1AHTR1DHTR1BDRD2HTR2A
Hydrochloric Acid SCHEMBL4234312 0.77 HTR1A (0.45) HTR1AHTR1DHTR1BDRD2HTR2A
SCHEMBL19280392 0.76 HSD11B1 (0.50) ALOX5HTR1AHTR1DHTR1BHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed