SCHEMBL4017563

SCHEMBL4017563

Oc1cccc(-c2ccnc3ccccc23)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.54
ACVR1 Q04771 4/20 0.50
FYN P06241 1/20 0.50
CDC7 O00311 1/20 0.50
TLR8 Q9NR97 1/20 0.49
CCNB2 O95067 1/20 0.49
CDK1 P06493 1/20 0.49
CCNB1 P14635 1/20 0.49
CCNB3 Q8WWL7 1/20 0.49
NPC1 O15118 1/20 0.48
ESR1 P03372 1/20 0.48
TP53 P04637 1/20 0.48
MAPT P10636 1/20 0.48
RAB9A P51151 1/20 0.48
PTK2B Q14289 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
AURKA O14965 1/20 0.47
TTK P33981 1/20 0.47
AURKB Q96GD4 1/20 0.47
INCENP Q9NQS7 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19991864 0.83 PIK3CA (0.59) ACVR1NPC1RAB9AAURKATTK
SCHEMBL30583075 0.83 PIK3CA (0.59) ACVR1NPC1RAB9AAURKATTK
SCHEMBL27433308 0.82 ACVR1 (0.52) ACVR1TLR8NPC1ESR1TP53
SCHEMBL27278122 0.81 BMP4 (0.57) ACVR1TLR8NPC1ESR1TP53
SCHEMBL28659657 0.80 GRM4 (0.61) ACVR1CDC7MAPTRAB9AAURKA
SCHEMBL14320615 0.80 AURKA (0.54) ACVR1FYNNPC1RAB9AAURKA
SCHEMBL21982345 0.80 ACVR1 (0.52) ACVR1NPC1MAPTRAB9AAURKA
SCHEMBL28647085 0.80 NUDT1 (0.57) ACVR1TLR8AURKATTKAURKB
SCHEMBL35327 0.80 TGFBR1 (0.60) ACVR1NPC1ESR1TP53MAPT
SCHEMBL30439957 0.80 TGFBR1 (0.60) ACVR1NPC1ESR1TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101541751-A Quinoline compounds WYETH CORP (US) 2009-09-23 CN disclosed
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed