SCHEMBL4017672

SCHEMBL4017672

CCCC(=O)C(Cc1ccc(-c2ccccc2C#N)cc1Cl)C(=O)OCC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F10 P00742 1/20 0.38
PPARG P37231 3/20 0.36
GRIA2 P42262 1/20 0.36
GRIA4 P48058 1/20 0.36
HSD17B3 P37058 1/20 0.36
MME P08473 1/20 0.35
CTSA P10619 2/20 0.35
ALDH1A1 P00352 2/20 0.35
GAA P10253 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C9 P11712 1/20 0.35
FFAR1 O14842 1/20 0.35
AKR1B1 P15121 1/20 0.35
CYP1A2 P05177 1/20 0.35
ALOX15 P16050 1/20 0.35
CYP2C19 P33261 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
AGTR1 P30556 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1369868 0.88 ALOX5AP (0.42) GRIA2GRIA4MMECTSAALDH1A1
SCHEMBL1372453 0.87 AGTR1 (0.45) F10GRIA2GRIA4ALDH1A1L3MBTL1
SCHEMBL1369710 0.86 AR (0.43) PPARG
SCHEMBL27962068 0.83 MME (0.47) PPARGGRIA2GRIA4MMEALDH1A1
SCHEMBL1370358 0.83 MME (0.47) PPARGGRIA2GRIA4MMEALDH1A1
SCHEMBL9846013 0.83 TSHR (0.36) PPARGGRIA2GRIA4MMECTSA
SCHEMBL1896656 0.81 RORC (0.37) PPARGMMEALDH1A1GAAL3MBTL1
SCHEMBL1895025 0.78 MME (0.46) PPARGGRIA2GRIA4MMEALDH1A1
SCHEMBL9845999 0.77 FFAR1 (0.41) MMECTSAALDH1A1GAAL3MBTL1
SCHEMBL1374269 0.77 MMP8 (0.38) PPARGMMEALDH1A1GAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009133970-A1 CRYSTALLINE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-05 WO disclosed
EP-2074117-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008062905-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-29 WO disclosed