SCHEMBL4019648

SCHEMBL4019648

CC(=O)Cc1ncc(Cl)nc1Cl

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 8/20 0.35
ALDH1A1 P00352 3/20 0.33
TDP1 Q9NUW8 2/20 0.33
SIRT6 Q8N6T7 1/20 0.32
PDCD1 Q15116 1/20 0.31
CD274 Q9NZQ7 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
AGBL2 Q5U5Z8 1/20 0.31
MAPK1 P28482 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28048176 0.83 AGBL2 (0.42) MAPKAPK2ALDH1A1TDP1SIRT6PDCD1
SCHEMBL17908109 0.79 S1PR2 (0.32) MAPKAPK2ALDH1A1TDP1SIRT6PDCD1
SCHEMBL31373452 0.77 MAPKAPK2 (0.46) MAPKAPK2
SCHEMBL17423463 0.77 MAPKAPK2 (0.46) MAPKAPK2
SCHEMBL12130919 0.75 MAPKAPK2 (0.33) MAPKAPK2ALDH1A1PDCD1CD274
SCHEMBL17908105 0.75 GRIK1 (0.36) TDP1
SCHEMBL26046044 0.75 PDE4A (0.34) TDP1NPC1RAB9AKMT2ASMN1; SMN2
SCHEMBL30529535 0.74 PDXK (0.35) MAPKAPK2ALDH1A1PDCD1CD274
SCHEMBL13259944 0.74 ALDH1A1 (0.38) MAPKAPK2ALDH1A1TDP1PDCD1CD274
SCHEMBL19641414 0.74 PDXK (0.35) MAPKAPK2ALDH1A1PDCD1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009089042-A1 PYRAZOLE PYRAZINE AMINE COMPOUNDS AS KINASE INHIBITORS, COMPOSITIONS THEREOF AND METHODS OF TREATMENT THEREWITH SIGNAL PHARMACEUTICALS, LLC (US) 2009-07-16 WO disclosed