SCHEMBL4021763

SCHEMBL4021763

COc1cccc(C(=O)C2CN(C(=O)C(C)(C)CCNC(=O)OC(C)(C)C)CC(C(=O)c3cccc(OC)c3)C2c2cccc(F)c2C)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.37
THRB P10828 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
KDM2B Q8NHM5 3/20 0.36
CHRM1 P11229 1/20 0.36
KMT2A Q03164 2/20 0.35
HTT P42858 1/20 0.35
DRD4 P21917 2/20 0.35
DRD2 P14416 1/20 0.35
MEN1 O00255 1/20 0.35
GFER P55789 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
HSD17B10 Q99714 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
HSD11B1 P28845 1/20 0.35
RAB9A P51151 2/20 0.34
ALDH1A1 P00352 1/20 0.34
OPRM1 P35372 1/20 0.34
NAMPT P43490 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13720836 1.00 SMN1; SMN2 (0.37) SMN1; SMN2THRBRXFP1KDM2BCHRM1
SCHEMBL4021768 1.00 SMN1; SMN2 (0.37) SMN1; SMN2THRBRXFP1KDM2BCHRM1
SCHEMBL4022167 0.89 DRD4 (0.42) SMN1; SMN2THRBRXFP1KDM2BDRD4
SCHEMBL13721566 0.89 DRD4 (0.42) SMN1; SMN2THRBRXFP1KDM2BDRD4
SCHEMBL4022160 0.89 DRD4 (0.42) SMN1; SMN2THRBRXFP1KDM2BDRD4
SCHEMBL4752775 0.87 DRD2 (0.46) DRD4DRD2
SCHEMBL4749499 0.87 DRD2 (0.45) DRD4DRD2
SCHEMBL13721648 0.85 HSD11B1 (0.38) SMN1; SMN2KDM2BKMT2AHTTMEN1
SCHEMBL5635169 0.82 KMT2A (0.37) SMN1; SMN2KDM2BKMT2AHTTMEN1
SCHEMBL5635174 0.82 KMT2A (0.37) SMN1; SMN2KDM2BKMT2AHTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7572814-B2 3,5-dibenzoyl-4-phenyl-piperidine anti-cancer compounds CYTOKINETICS, INCORPORATED (US) 2009-08-11 US disclosed
EP-1962846-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-09-03 EP disclosed
WO-2007059323-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-24 WO disclosed