SCHEMBL4021824

SCHEMBL4021824

CC(C)(CN)OC(=O)N1CCCCC1c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 5/20 0.56
TMEM97 Q5BJF2 4/20 0.46
SIGMAR1 Q99720 4/20 0.46
HSD11B1 P28845 1/20 0.46
PRMT5 O14744 4/20 0.45
WDR77 Q9BQA1 4/20 0.45
PARP14 Q460N5 1/20 0.45
PARP10 Q53GL7 1/20 0.45
EPHX2 P34913 2/20 0.43
HSP90AA1 P07900 1/20 0.42
HSP90AB1 P08238 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24365782 0.85 RIPK1 (0.63) RIPK1TMEM97SIGMAR1HSD11B1PRMT5
SCHEMBL7469150 0.85 RIPK1 (0.63) RIPK1TMEM97SIGMAR1HSD11B1PRMT5
SCHEMBL17114341 0.85 RIPK1 (0.63) RIPK1TMEM97SIGMAR1HSD11B1PRMT5
Water SCHEMBL27902502 0.84 RIPK1 (0.62) RIPK1TMEM97SIGMAR1HSD11B1PRMT5
SCHEMBL30281143 0.84 RIPK1 (0.62) RIPK1TMEM97SIGMAR1HSD11B1PRMT5
SCHEMBL27830000 0.82 RIPK1 (0.59) RIPK1TMEM97SIGMAR1HSD11B1PRMT5
SCHEMBL6960066 0.81 RIPK1 (0.69) RIPK1EPHX2HSP90AA1HSP90AB1
SCHEMBL18642714 0.81 RIPK1 (0.69) RIPK1EPHX2HSP90AA1HSP90AB1
SCHEMBL8303313 0.80 TMEM97 (0.58) RIPK1TMEM97SIGMAR1HSD11B1PRMT5
SCHEMBL4277144 0.80 RIPK1 (0.59) RIPK1TMEM97SIGMAR1HSD11B1PRMT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1545525-A4 RADIOLABELED NEUROKININ-1 RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2009-07-01 EP disclosed
EP-1119356-A4 RADIOLABELED NEUROKININ-1 RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2008-01-09 EP disclosed
EP-1545525-A2 RADIOLABELED NEUROKININ-1 RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2005-06-29 EP disclosed
WO-2004029024-A2 RADIOLABELED NEUROKININ-1 RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2004-04-08 WO disclosed
EP-1119356-A1 RADIOLABELED NEUROKININ-1 RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2001-08-01 EP disclosed
WO-2000018403-A1 RADIOLABELED NEUROKININ-1 RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2000-04-06 WO disclosed