SCHEMBL4022840

SCHEMBL4022840

O=C(O)NC(CO)c1ncc(F)cc1F

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AGBL2 Q5U5Z8 1/20 0.39
MAPK1 P28482 8/20 0.35
CNR2 P34972 2/20 0.34
PTGER4 P35408 1/20 0.33
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
PPARG P37231 1/20 0.32
S1PR1 P21453 3/20 0.32
S1PR3 Q99500 3/20 0.32
GPR88 Q9GZN0 1/20 0.32
ROCK2 O75116 2/20 0.31
ROCK1 Q13464 1/20 0.31
S1PR2 O95136 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL590718 0.83 AGBL2 (0.38) AGBL2PTGER4CYP1A2CYP3A4CYP2D6
SCHEMBL588556 0.83 AGBL2 (0.38) AGBL2PTGER4CYP1A2CYP3A4CYP2D6
SCHEMBL4019098 0.83 MAPK1 (0.39) AGBL2MAPK1PTGER4
SCHEMBL3947856 0.74 APLNR (0.39) AGBL2MAPK1
SCHEMBL588356 0.69 L3MBTL1 (0.43) PTGER4
SCHEMBL896777 0.69 AKR1C3 (0.44) AGBL2PTGER4CYP1A2CYP3A4CYP2D6
SCHEMBL588357 0.69 L3MBTL1 (0.43) PTGER4
SCHEMBL3944958 0.69 AGBL2 (0.38) AGBL2MAPK1PTGER4CYP2D6CYP2C19
SCHEMBL12985296 0.68 MEN1 (0.44) AGBL2MAPK1CYP1A2CYP3A4CYP2C19
SCHEMBL4070072 0.67 CNR2 (0.45) MAPK1CNR2GPR88ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009016410-A2 CHEMICAL COMPOUNDS 831 ASTRAZENECA AB (SE) 2009-02-05 WO disclosed
WO-2008132502-A1 PYRAZOLYL-AMINO-SUBSTITUTED PYRIMIDINES AND THEIR USE FOR THE TREATMENT OF CANCER ASTRAZENECA AB (SE) 2008-11-06 WO disclosed