SCHEMBL4024212

SCHEMBL4024212

O=C(O)C(C(=O)C1CCC(C(F)(F)F)CC1)c1ccc2ocnc2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
KMT2A Q03164 1/20 0.38
CTNNB1 P35222 3/20 0.36
WNT3A P56704 3/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
FABP4 P15090 1/20 0.33
BRD4 O60885 1/20 0.31
CREBBP Q92793 1/20 0.31
TBK1 Q9UHD2 1/20 0.31
ESR1 P03372 1/20 0.31
NAMPT P43490 1/20 0.30
PDE4A P27815 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4C Q08493 1/20 0.30
PDE4D Q08499 1/20 0.30
FASN P49327 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13746010 0.88 BRD4 (0.34) MEN1ALDH1A1GAAKMT2ACTNNB1
SCHEMBL4021493 0.74 KDM4E (0.38) MEN1GAAKMT2ASMN1; SMN2
SCHEMBL4020465 0.65 HSD17B10 (0.45) MEN1ALDH1A1GAAKMT2ANPC1
SCHEMBL24865700 0.65 ULK1 (0.37) ALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL30336302 0.65 ULK1 (0.37) ALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL13746955 0.62 PI4KB (0.36) MEN1ALDH1A1GAAKMT2ANPC1
SCHEMBL8007655 0.62 SRC (0.61) MEN1ALDH1A1GAAKMT2A
Trifluoroacetic Acid SCHEMBL29479758 0.62 MEN1 (0.50) MEN1ALDH1A1GAAKMT2ACTNNB1
SCHEMBL4025663 0.61 DPP4 (0.38) ALDH1A1KMT2A
SCHEMBL31003292 0.61 MEN1 (0.45) MEN1ALDH1A1GAAKMT2ACTNNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100403-A1 SUBSTITUTED ARYL PYRIMIDINONES NEUROGEN CORPORATION (US) 2009-08-13 WO disclosed