SCHEMBL4024508

SCHEMBL4024508

OCc1ccc(N2CCNCC2)cn1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 8/20 0.58
CHRNA4 P43681 8/20 0.58
AOC3 Q16853 1/20 0.53
ADRB1 P08588 3/20 0.44
HRH3 Q9Y5N1 2/20 0.44
HTR3E A5X5Y0 2/20 0.44
HTR3B O95264 2/20 0.44
HTR3A P46098 2/20 0.44
HTR3D Q70Z44 2/20 0.44
HTR3C Q8WXA8 2/20 0.44
SIGMAR1 Q99720 2/20 0.44
KDM4E B2RXH2 1/20 0.44
ADRB2 P07550 1/20 0.44
NCF1 P14598 1/20 0.44
PLD1 Q13393 1/20 0.44
CDK4 P11802 1/20 0.43
CCND1 P24385 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12147196 0.83 CHRNB2 (0.58) CHRNB2CHRNA4AOC3ADRB1HTR3E
SCHEMBL22876928 0.81 CHRNB2 (0.57) CHRNB2CHRNA4AOC3ADRB1HTR3E
SCHEMBL30922297 0.80 CHKA (0.51) HRH3HTR3AKDM4E
SCHEMBL3650490 0.80 POLB (0.51) HRH3KDM4E
SCHEMBL25376115 0.80 CHRNB2 (0.54) CHRNB2CHRNA4AOC3ADRB1HTR3E
SCHEMBL14341117 0.80 CHRNB2 (0.54) CHRNB2CHRNA4AOC3ADRB1HTR3E
SCHEMBL31058076 0.79 WNT3A (0.45) CHRNB2CHRNA4AOC3HRH3KDM4E
SCHEMBL31073166 0.79 HRH3 (0.44) AOC3HRH3
SCHEMBL22411598 0.77 CHRNB2 (0.64) CHRNB2CHRNA4ADRB1HTR3EHTR3B
SCHEMBL3853696 0.76 HRH3 (0.53) AOC3HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1718307-A4 IMMUNOSUPPRESSANT COMPOUNDS AND COMPOSITIONS IRM LLC (BM) 2009-04-29 EP disclosed
EP-1718307-A2 IMMUNOSUPPRESSANT COMPOUNDS AND COMPOSITIONS IRM, LLC (BM) 2006-11-08 EP disclosed
WO-2005082089-A2 IMMUNOSUPPRESSANT COMPOUNDS AND COMPOSITIONS IRM LLC (BM) 2005-09-09 WO disclosed