SCHEMBL4025213

SCHEMBL4025213

CC(=O)c1cccc(-c2ccc3nc(-c4cccc(F)c4)cc(N(C)C)c3c2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.44
KDM1A O60341 1/20 0.44
MAP4K4 O95819 2/20 0.44
CSNK1G2 P78368 2/20 0.44
CLK4 Q9HAZ1 2/20 0.44
MKNK2 Q9HBH9 2/20 0.44
MAP4K5 Q9Y4K4 2/20 0.44
DHODH Q02127 2/20 0.43
NT5E P21589 2/20 0.43
AURKA O14965 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ACP1 P24666 1/20 0.40
CDK2 P24941 2/20 0.40
PLK4 O00444 1/20 0.40
DCLK1 O15075 1/20 0.40
ROCK2 O75116 1/20 0.40
PRKD3 O94806 1/20 0.40
PAK4 O96013 1/20 0.40
CHEK2 O96017 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4031738 0.86 DHODH (0.45) MAP4K4CLK4DHODHNT5EMEN1
SCHEMBL4026356 0.84 NT5E (0.43) MAP4K4DHODHNT5EMEN1KMT2A
SCHEMBL4027654 0.81 ACP1 (0.48) CLK4DHODHNT5EAURKAMEN1
SCHEMBL4022559 0.81 NT5E (0.49) MAP4K4DHODHNT5EACP1CDK2
SCHEMBL4025761 0.80 NT5E (0.44) MAP4K4DHODHNT5EMEN1KMT2A
SCHEMBL4823424 0.79 MAP4K4 (0.43) MAP4K4DHODHNT5EMEN1KMT2A
SCHEMBL4025078 0.79 RXFP1 (0.42) MAP4K4KMT2AACP1
SCHEMBL4032316 0.79 CYP1A2 (0.46) CLK4DHODHNT5EACP1KDR
SCHEMBL4026216 0.78 FYN (0.46) KDM1ANT5EMEN1KMT2AACP1
SCHEMBL4031533 0.78 LMNA (0.47) CLK4DHODHMEN1KMT2ACLK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339690-B1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2009-01-21 EP disclosed