SCHEMBL4031533

SCHEMBL4031533

CN(C)c1cc(-c2cccc(F)c2)nc2ccc(-c3ccc4c(c3)OCO4)cc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.47
ALDH1A1 P00352 5/20 0.47
CLK4 Q9HAZ1 4/20 0.47
HSD17B10 Q99714 4/20 0.47
CYP1A2 P05177 3/20 0.47
CYP3A4 P08684 3/20 0.47
CYP2D6 P10635 3/20 0.47
CYP2C19 P33261 3/20 0.47
TSHR P16473 3/20 0.47
MAPK1 P28482 3/20 0.47
HIF1A Q16665 1/20 0.47
KMT2A Q03164 5/20 0.46
TP53 P04637 2/20 0.46
CYP2C9 P11712 2/20 0.46
USP2 O75604 1/20 0.46
ALOX15 P16050 1/20 0.46
DHODH Q02127 1/20 0.46
ADORA2A P29274 2/20 0.46
ADORA1 P30542 2/20 0.46
CLK1 P49759 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4031738 0.84 DHODH (0.45) CLK4KMT2ADHODHADORA2AMEN1
SCHEMBL4029317 0.84 CLK4 (0.48) LMNAALDH1A1CLK4HSD17B10CYP1A2
SCHEMBL4026356 0.82 NT5E (0.43) ALDH1A1KMT2AALOX15DHODHADORA2A
SCHEMBL4027654 0.79 ACP1 (0.48) LMNAALDH1A1CLK4CYP1A2CYP3A4
SCHEMBL4022559 0.79 NT5E (0.49) DHODHTDP1
SCHEMBL4025213 0.78 DHFR (0.44) CLK4KMT2ADHODHMEN1CLK2
SCHEMBL4025761 0.78 NT5E (0.44) KMT2ADHODHADORA2AKDM4EMEN1
SCHEMBL4025078 0.77 RXFP1 (0.42) KMT2AADORA2AKDM4EGAAHPGD
SCHEMBL4823424 0.77 MAP4K4 (0.43) LMNAALDH1A1KMT2ADHODHADORA2A
SCHEMBL4032316 0.77 CYP1A2 (0.46) LMNAALDH1A1CLK4CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339690-B1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2009-01-21 EP disclosed