SCHEMBL4026490

SCHEMBL4026490

COC(=O)C1CCCCN1C(=O)C1CN(CCN(C)S(C)(=O)=O)CC(C(=O)c2cccc(O)c2)C1c1cccc(F)c1C

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.34
TSHR P16473 1/20 0.34
GALR3 O60755 1/20 0.33
NR2F2 P24468 1/20 0.33
RAB9A P51151 1/20 0.33
LOX P28300 1/20 0.33
F2 P00734 2/20 0.31
PLG P00747 2/20 0.31
ST14 Q9Y5Y6 2/20 0.31
F10 P00742 1/20 0.31
PLAU P00749 1/20 0.31
SCN9A Q15858 1/20 0.31
GAA P10253 1/20 0.30
PDCD1 Q15116 1/20 0.30
CD274 Q9NZQ7 1/20 0.30
FKBP1A P62942 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4025921 1.00 ALDH1A1 (0.34) ALDH1A1CYP3A4TSHRGALR3NR2F2
SCHEMBL4027055 0.98 ALDH1A1 (0.36) ALDH1A1CYP3A4TSHRGALR3NR2F2
SCHEMBL4019629 0.98 ALDH1A1 (0.36) ALDH1A1CYP3A4TSHRGALR3NR2F2
SCHEMBL4752899 0.90 GYS1 (0.34)
SCHEMBL4752900 0.90 GYS1 (0.34)
SCHEMBL4022158 0.86 BCHE (0.31) SCN9A
SCHEMBL4021872 0.86 BCHE (0.31) SCN9A
SCHEMBL4028041 0.86 OPRM1 (0.35)
SCHEMBL4028045 0.86 OPRM1 (0.35)
SCHEMBL13721487 0.86 OPRM1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7572814-B2 3,5-dibenzoyl-4-phenyl-piperidine anti-cancer compounds CYTOKINETICS, INCORPORATED (US) 2009-08-11 US disclosed