SCHEMBL4028883

SCHEMBL4028883

O=C(CCl)C1CCN(C(=O)O)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
YAP1 P46937 1/20 0.41
TEAD4 Q15561 1/20 0.41
MAPT P10636 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
LMNA P02545 2/20 0.34
GAA P10253 1/20 0.34
RAB9A P51151 2/20 0.34
ABL1 P00519 1/20 0.33
RIN1 Q13671 1/20 0.33
POLB P06746 1/20 0.33
NPC1 O15118 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MEN1 O00255 1/20 0.33
TSHR P16473 1/20 0.33
KMT2A Q03164 1/20 0.33
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11882770 0.83 ALDH1A1 (0.62) ALDH1A1YAP1TEAD4L3MBTL1LMNA
SCHEMBL12359795 0.82 ALDH1A1 (0.46) ALDH1A1LMNAGAASMN1; SMN2
SCHEMBL17713778 0.79 GAA (0.42) ALDH1A1MAPTL3MBTL1LMNAGAA
SCHEMBL1535175 0.79 NLRP3 (0.36) ALDH1A1MAPTL3MBTL1LMNAGAA
SCHEMBL146591 0.77 MAPT (0.37) ALDH1A1YAP1TEAD4MAPTL3MBTL1
SCHEMBL13714198 0.77 ALDH1A1 (0.39) ALDH1A1LMNAABL1RIN1SMN1; SMN2
SCHEMBL1132078 0.77
SCHEMBL31348822 0.76 ABL1 (0.44) ALDH1A1MAPTLMNAGAAABL1
SCHEMBL14854942 0.76 L3MBTL1 (0.33) MAPTL3MBTL1LMNAGAARAB9A
SCHEMBL5184241 0.76 MAPT (0.38) ALDH1A1YAP1TEAD4MAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061759-A1 CYCLIC MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Brystol-Myers Squibb Company (US) 2009-05-27 EP disclosed
WO-2008042926-A1 CYCLIC MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL-MYERS SQUIBB COMPANY (US) 2008-04-10 WO disclosed