SCHEMBL4029417

SCHEMBL4029417

Cc1onc(-c2cccc(C(F)(F)F)c2)c1NC(=O)O

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 1/20 0.53
NTRK1 P04629 2/20 0.53
EPAS1 Q99814 3/20 0.49
MAPT P10636 3/20 0.47
POLB P06746 2/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
LMNA P02545 1/20 0.46
MAPK1 P28482 1/20 0.46
TSHR P16473 2/20 0.46
HTT P42858 1/20 0.45
BRD4 O60885 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
IP6K1 Q92551 1/20 0.45
IP6K3 Q96PC2 1/20 0.45
IP6K2 Q9UHH9 1/20 0.45
ALDH1A1 P00352 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
XDH P47989 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4032643 0.83 TSHR (0.51) GPBAR1NTRK1MAPTKMT2ATSHR
SCHEMBL13733019 0.82 GPBAR1 (0.64) GPBAR1EPAS1MAPTPOLBMEN1
SCHEMBL4029460 0.81 NPSR1 (0.61) NTRK1MAPTMEN1KMT2AMAPK1
SCHEMBL4034243 0.81 KMT2A (0.49) NTRK1MAPTMEN1KMT2ATSHR
SCHEMBL11420447 0.79 GPBAR1 (0.61) GPBAR1EPAS1MAPTPOLBMEN1
SCHEMBL27936782 0.79 GPBAR1 (0.53) GPBAR1EPAS1MAPTPOLBBRD4
SCHEMBL13734246 0.79 GPBAR1 (0.61) GPBAR1EPAS1MAPTPOLBMEN1
SCHEMBL4033713 0.78 LPAR1 (0.48) GPBAR1NTRK1EPAS1KMT2A
SCHEMBL5777101 0.77 RXRA (0.54) GPBAR1MAPTBRD4IP6K1IP6K3
SCHEMBL27936779 0.77 GPBAR1 (0.55) GPBAR1EPAS1MAPTPOLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1258484-B1 NOVEL ISOXAZOLE AND THIAZOLE COMPOUNDS AND USE THEREOF AS DRUGS KYOWA HAKKO KIRIN CO LTD (JP) 2009-01-14 EP claimed