SCHEMBL4034243

SCHEMBL4034243

Cc1onc(-c2cccc(Br)c2)c1NC(=O)O

nearest known ligand 0.62

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.49
CACNA1F O60840 1/20 0.48
ABCB1 P08183 1/20 0.48
CACNA1D Q01668 1/20 0.48
CACNA1S Q13698 1/20 0.48
CACNA1C Q13936 1/20 0.48
TSHR P16473 1/20 0.48
HTT P42858 1/20 0.48
NPSR1 Q6W5P4 2/20 0.47
ALDH1A1 P00352 4/20 0.46
TDP1 Q9NUW8 1/20 0.46
MAPT P10636 2/20 0.46
KDM4E B2RXH2 1/20 0.45
NTRK1 P04629 2/20 0.45
ALOX12 P18054 1/20 0.44
GAA P10253 2/20 0.43
MEN1 O00255 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4029460 0.84 NPSR1 (0.61) KMT2ATSHRHTTNPSR1ALDH1A1
SCHEMBL4032643 0.84 TSHR (0.51) KMT2ATSHRHTTNPSR1ALDH1A1
SCHEMBL9903838 0.83 NPSR1 (0.48) KMT2ACACNA1FABCB1CACNA1DCACNA1S
SCHEMBL4029417 0.81 GPBAR1 (0.53) KMT2ATSHRHTTNPSR1ALDH1A1
SCHEMBL2473629 0.78 KMT2A (0.51) KMT2ACACNA1FABCB1CACNA1DCACNA1S
SCHEMBL4033731 0.78 LPAR1 (0.51) KMT2ANPSR1MAPTGAA
SCHEMBL4037282 0.77 MAPT (0.52) KMT2ATSHRHTTNPSR1ALDH1A1
SCHEMBL2470464 0.75 CACNA1F (0.50) KMT2ACACNA1FABCB1CACNA1DCACNA1S
SCHEMBL4028725 0.74 MAPT (0.49) KMT2ATSHRHTTNPSR1ALDH1A1
SCHEMBL5527223 0.74 MEN1 (0.61) KMT2ATSHRHTTNPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1258484-B1 NOVEL ISOXAZOLE AND THIAZOLE COMPOUNDS AND USE THEREOF AS DRUGS KYOWA HAKKO KIRIN CO LTD (JP) 2009-01-14 EP claimed