SCHEMBL4030241

SCHEMBL4030241

Cc1noc(-c2ccc(CNCCc3ccccn3)cc2)c1N(C(=O)O)C(C)c1ccccc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LPAR1 Q92633 3/20 0.42
LPAR2 Q9HBW0 2/20 0.42
LPAR3 Q9UBY5 2/20 0.42
HTR5A P47898 1/20 0.40
ALDH1A1 P00352 3/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C19 P33261 1/20 0.37
TDP1 Q9NUW8 1/20 0.36
LMNA P02545 1/20 0.36
PKM P14618 1/20 0.36
SLC12A2 P55011 1/20 0.36
SLC12A5 Q9H2X9 1/20 0.36
NR3C2 P08235 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
CD274 Q9NZQ7 1/20 0.35
NMT1 P30419 1/20 0.35
KDM4E B2RXH2 2/20 0.35
NR3C1 P04150 1/20 0.34
HTT P42858 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4028841 0.93 LPAR1 (0.43) LPAR1LPAR2LPAR3ALDH1A1CYP1A2
SCHEMBL4036454 0.89 LPAR1 (0.43) LPAR1LPAR2LPAR3HTR5AALDH1A1
SCHEMBL4034939 0.87 LPAR1 (0.45) LPAR1LPAR2LPAR3HTR5AALDH1A1
SCHEMBL4031158 0.87 MEN1 (0.43) LPAR1LPAR2LPAR3HTR5AALDH1A1
SCHEMBL4032394 0.86 LPAR1 (0.47) LPAR1LPAR2LPAR3KDM4E
SCHEMBL4036696 0.85 LPAR1 (0.44) LPAR1LPAR2LPAR3KDM4E
SCHEMBL4032920 0.82 ATM (0.44) LPAR1LPAR2LPAR3ALDH1A1TDP1
SCHEMBL4034499 0.81 LPAR1 (0.48) LPAR1LPAR2LPAR3ALDH1A1KDM4E
SCHEMBL4034108 0.80 LPAR1 (0.44) LPAR1LPAR2LPAR3ALDH1A1LMNA
SCHEMBL4034918 0.80 LPAR1 (0.45) LPAR1LPAR2LPAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1258484-B1 NOVEL ISOXAZOLE AND THIAZOLE COMPOUNDS AND USE THEREOF AS DRUGS KYOWA HAKKO KIRIN CO LTD (JP) 2009-01-14 EP claimed