SCHEMBL4031154

SCHEMBL4031154

CCc1noc(-c2ccc(C#N)cc2)c1NC(=O)O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
PKM P14618 1/20 0.41
TRPA1 O75762 1/20 0.41
TP53 P04637 3/20 0.39
LMNA P02545 2/20 0.39
MAPT P10636 2/20 0.39
RXFP1 Q9HBX9 1/20 0.38
DHODH Q02127 1/20 0.37
GRIA2 P42262 1/20 0.37
GRIA4 P48058 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
KDM4E B2RXH2 1/20 0.36
GSK3B P49841 1/20 0.36
SCD O00767 1/20 0.36
EGLN1 Q9GZT9 1/20 0.36
PPARG P37231 1/20 0.36
PPARD Q03181 1/20 0.36
PPARA Q07869 1/20 0.36
THRB P10828 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4027976 0.85 MAPT (0.49) ALDH1A1PKMTRPA1TP53LMNA
SCHEMBL4034308 0.84 KDM4E (0.49) ALDH1A1LMNAMAPTSMN1; SMN2KDM4E
SCHEMBL4304 0.83 RAB9A (0.40) ALDH1A1TP53MAPTRXFP1SMN1; SMN2
SCHEMBL4033611 0.81 LPAR1 (0.40) ALDH1A1TP53MAPTSMN1; SMN2KDM4E
SCHEMBL4029624 0.77 LPAR1 (0.59)
SCHEMBL13960108 0.75 CYP2A6 (0.41) TP53LMNAMAPTDHODHKDM4E
SCHEMBL3704614 0.71 TRPA1 (0.56) ALDH1A1PKMTRPA1TP53LMNA
SCHEMBL15464353 0.71 PTPN1 (0.45) ALDH1A1PKMTRPA1TP53LMNA
SCHEMBL4036888 0.71 LPAR1 (0.47) ALDH1A1LMNAMAPTKDM4E
SCHEMBL15013106 0.71 LPAR1 (0.50) ALDH1A1TRPA1MAPTSMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1258484-B1 NOVEL ISOXAZOLE AND THIAZOLE COMPOUNDS AND USE THEREOF AS DRUGS KYOWA HAKKO KIRIN CO LTD (JP) 2009-01-14 EP claimed