SCHEMBL4032705

SCHEMBL4032705

Cc1onc(-c2cccc(F)c2)c1N(C(=O)O)C(C)c1ccccc1Cl

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.48
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
GAA P10253 2/20 0.42
ALDH1A1 P00352 2/20 0.42
MAPT P10636 2/20 0.42
LMNA P02545 1/20 0.42
KDM4E B2RXH2 1/20 0.40
PPARG P37231 1/20 0.40
NCOA2 Q15596 1/20 0.40
GABRA5 P31644 2/20 0.40
CTSA P10619 1/20 0.40
PTGS2 P35354 2/20 0.39
PTGS1 P23219 1/20 0.39
TSHR P16473 1/20 0.39
TP53 P04637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4029082 0.91 GAA (0.45) GPBAR1MEN1KMT2AGAAALDH1A1
SCHEMBL4028916 0.91 GAA (0.45) GPBAR1MEN1KMT2AGAAALDH1A1
SCHEMBL4034254 0.90 KMT2A (0.44) GPBAR1MEN1KMT2AGAAALDH1A1
SCHEMBL4037046 0.89 KMT2A (0.43) GPBAR1MEN1KMT2AGAAALDH1A1
SCHEMBL4034655 0.89 GPBAR1 (0.49) GPBAR1MEN1KMT2AGAAALDH1A1
SCHEMBL4029400 0.85 ALDH1A1 (0.43) GPBAR1MEN1KMT2AGAAALDH1A1
SCHEMBL4030964 0.84 HDAC3 (0.39) GPBAR1MEN1KMT2AGAAALDH1A1
SCHEMBL4032656 0.84 MEN1 (0.48) GPBAR1MEN1KMT2AGAAALDH1A1
SCHEMBL4033798 0.82 MEN1 (0.43) GPBAR1MEN1KMT2AGAAALDH1A1
SCHEMBL4036403 0.82 NPSR1 (0.45) MEN1KMT2AGAAALDH1A1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1258484-B1 NOVEL ISOXAZOLE AND THIAZOLE COMPOUNDS AND USE THEREOF AS DRUGS KYOWA HAKKO KIRIN CO LTD (JP) 2009-01-14 EP claimed