SCHEMBL4037046

SCHEMBL4037046

Cc1onc(-c2cccc(Br)c2)c1N(C(=O)O)C(C)c1ccccc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.43
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
MEN1 O00255 1/20 0.40
CACNA1F O60840 1/20 0.39
ABCB1 P08183 1/20 0.39
CACNA1D Q01668 1/20 0.39
CACNA1S Q13698 1/20 0.39
CACNA1C Q13936 1/20 0.39
PTGS2 P35354 2/20 0.39
PTGFR P43088 6/20 0.39
PTGS1 P23219 1/20 0.38
NPSR1 Q6W5P4 2/20 0.38
RORB Q92753 1/20 0.38
GPBAR1 Q8TDU6 1/20 0.38
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4029082 0.90 GAA (0.45) KMT2AALDH1A1LMNAGAAMAPT
SCHEMBL4028916 0.90 GAA (0.45) KMT2AALDH1A1LMNAGAAMAPT
SCHEMBL4032705 0.89 GPBAR1 (0.48) KMT2AALDH1A1LMNAGAAMAPT
SCHEMBL4034655 0.86 GPBAR1 (0.49) KMT2AALDH1A1LMNAGAAMAPT
SCHEMBL4029400 0.85 ALDH1A1 (0.43) KMT2AALDH1A1LMNAGAAMAPT
SCHEMBL4034254 0.83 KMT2A (0.44) KMT2AALDH1A1LMNAGAAMAPT
SCHEMBL4033798 0.81 MEN1 (0.43) KMT2AALDH1A1LMNAGAAMAPT
SCHEMBL4034797 0.81 NPSR1 (0.45) KMT2AALDH1A1GAAMEN1PTGS2
SCHEMBL4028127 0.81 NPSR1 (0.45) KMT2AALDH1A1GAAMEN1PTGS2
SCHEMBL4033782 0.80 MAPK1 (0.42) KMT2AALDH1A1LMNAGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1258484-B1 NOVEL ISOXAZOLE AND THIAZOLE COMPOUNDS AND USE THEREOF AS DRUGS KYOWA HAKKO KIRIN CO LTD (JP) 2009-01-14 EP claimed