SCHEMBL4033591

SCHEMBL4033591

O=C(O)Cc1cccc(-c2cnco2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.58
CYP4A11 Q02928 1/20 0.58
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
MAP4K4 O95819 1/20 0.53
HDAC4 P56524 1/20 0.49
CYP11B1 P15538 1/20 0.45
CYP11B2 P19099 1/20 0.45
NAPRT Q6XQN6 1/20 0.45
GRIN2D O15399 1/20 0.45
GRIN3B O60391 1/20 0.45
GRIN1 Q05586 1/20 0.45
GRIN2A Q12879 1/20 0.45
GRIN2B Q13224 1/20 0.45
GRIN2C Q14957 1/20 0.45
GRIN3A Q8TCU5 1/20 0.45
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.44
NPC1 O15118 1/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3207637 0.81 MEN1 (0.58) MEN1KMT2AMAP4K4HDAC4CYP11B1
SCHEMBL29468019 0.78 MAP4K4 (0.63) MEN1KMT2AMAP4K4HDAC4CYP11B1
SCHEMBL3205366 0.78 MEN1 (0.63) CYP4F2CYP4A11MEN1KMT2AMAP4K4
SCHEMBL12298706 0.78 MEN1 (0.58) MEN1KMT2AMAP4K4HDAC4CYP11B1
SCHEMBL5664152 0.77 KEAP1 (0.59) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL940586 0.77 KEAP1 (0.59) MEN1KMT2AMAP4K4HDAC4CYP11B1
SCHEMBL2158739 0.77 KMT2A (0.75) MEN1KMT2AMAP4K4HDAC4CYP11B1
SCHEMBL10445828 0.76 KMT2A (0.49) CYP4F2CYP4A11MEN1KMT2AMAP4K4
SCHEMBL28032595 0.75 LMNA (0.63) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL22070661 0.74 CYP4F2 (1.00) CYP4F2CYP4A11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010493-A2 PYRIDYL AMIDE T-TYPE CALCIUM CHANNEL ANTAGONISTS Merck & Co., Inc. (US) 2009-01-07 EP disclosed
WO-2007120729-A2 PYRIDYL AMIDE T-TYPE CALCIUM CHANNEL ANTAGONISTS MERCK & CO., INC. (US) 2007-10-25 WO disclosed