SCHEMBL4033857

SCHEMBL4033857

CC(Cc1ccccc1)c1cccnc1CO

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
TRPA1 O75762 1/20 0.42
KMT2A Q03164 1/20 0.41
MAOA P21397 4/20 0.41
MAOB P27338 3/20 0.41
NISCH Q9Y2I1 3/20 0.41
KDM4E B2RXH2 1/20 0.41
TAAR1 Q96RJ0 4/20 0.40
SIGMAR1 Q99720 4/20 0.40
SLC18A2 Q05940 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4064147 0.79 ALDH1A1 (0.41) ALDH1A1L3MBTL1TRPA1KMT2AMAOA
SCHEMBL2084128 0.78 L3MBTL1 (0.53) ALDH1A1L3MBTL1KMT2ANISCHKDM4E
SCHEMBL4030522 0.74 TAAR1 (0.45) KMT2AMAOAMAOBNISCHKDM4E
SCHEMBL4033855 0.73 ALDH1A1 (0.44) ALDH1A1L3MBTL1CYP2D6NR3C2
SCHEMBL24313207 0.73 ALDH1A1 (0.41) ALDH1A1L3MBTL1KDM4ENPC1RAB9A
SCHEMBL4033860 0.72 ALDH1A1 (0.43) ALDH1A1L3MBTL1TRPA1MAOAMAOB
SCHEMBL8973031 0.71 L3MBTL1 (0.53) ALDH1A1L3MBTL1KMT2AKDM4ENPC1
SCHEMBL28115795 0.71 TAAR1 (0.52) TRPA1MAOATAAR1SIGMAR1SLC18A2
SCHEMBL1868728 0.71 TSHR (0.64) TRPA1MAOATAAR1SIGMAR1SLC18A2
SCHEMBL6547009 0.70 SIGMAR1 (0.52) TRPA1KMT2AMAOATAAR1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed