SCHEMBL4035655

SCHEMBL4035655

Cc1cccnc1CN(CCCCNC(=O)OC(C)(C)C)CC1(C(=O)OC(C)(C)C)Nc2ccccc2N1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.39
AKT1 P31749 2/20 0.38
PDPK1 O15530 1/20 0.37
CCNB2 O95067 1/20 0.37
PRKCB P05771 1/20 0.37
CDK1 P06493 1/20 0.37
LYN P07948 1/20 0.37
CCNB1 P14635 1/20 0.37
CCNA2 P20248 1/20 0.37
CDK2 P24941 1/20 0.37
GSK3B P49841 1/20 0.37
RPS6KA3 P51812 1/20 0.37
CCNA1 P78396 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37
CYP3A4 P08684 1/20 0.36
CKS1B P61024 1/20 0.36
SKP1 P63208 1/20 0.36
SKP2 Q13309 1/20 0.36
CXCR4 P61073 2/20 0.36
CHRM2 P08172 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2083428 0.82 CYP3A4 (0.43) DRD2CYP3A4CKS1BSKP1SKP2
SCHEMBL4032545 0.77 L3MBTL1 (0.40) DRD2PDPK1CCNB2PRKCBCDK1
SCHEMBL2081783 0.77 BCHE (0.48) CXCR4KDM4EBRD4
SCHEMBL4035412 0.76 DRD2 (0.42) DRD2CYP3A4CKS1BSKP1SKP2
SCHEMBL2086065 0.76 CXCR4 (0.41) DRD2PDPK1CCNB2PRKCBCDK1
SCHEMBL4032836 0.75 CXCR4 (0.40) DRD2PDPK1CCNB2PRKCBCDK1
SCHEMBL4039491 0.75 CYP3A4 (0.44) DRD2CYP3A4CKS1BSKP1SKP2
SCHEMBL2085099 0.74 BRD4 (0.46) CYP3A4BRD4ALDH1A1
SCHEMBL2084807 0.73 BRD4 (0.44) CYP3A4CXCR4KDM4EL3MBTL1BRD4
SCHEMBL2086066 0.72 CXCR4 (0.44) CYP3A4CXCR4KDM4EL3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed