SCHEMBL4034041

SCHEMBL4034041

O=C(c1ccc2c3c(ccc2c1)OCCC3)c1c[nH]cn1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
CTNNB1 P35222 3/20 0.34
WNT3A P56704 3/20 0.34
PIR O00625 2/20 0.33
HSF1 Q00613 2/20 0.33
HPGD P15428 2/20 0.33
TP53 P04637 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32
CHRNA7 P36544 2/20 0.32
MAPT P10636 2/20 0.32
KDM4E B2RXH2 1/20 0.32
USP2 O75604 1/20 0.32
ALDH1A1 P00352 1/20 0.32
RECQL P46063 1/20 0.32
HSD17B10 Q99714 1/20 0.32
POLB P06746 1/20 0.31
ATM Q13315 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4030413 0.93 NPC1 (0.32) NPC1RAB9ACTNNB1MTNR1AMTNR1B
SCHEMBL4024487 0.76 PRKCI (0.35) NPC1RAB9ACTNNB1WNT3ASMN1; SMN2
SCHEMBL4029004 0.74 NPC1 (0.37) NPC1RAB9ACTNNB1WNT3APIR
SCHEMBL4030416 0.73 CYP17A1 (0.31) MTNR1AMTNR1B
SCHEMBL4024232 0.71 CTNNB1 (0.33) RAB9ACTNNB1WNT3AHPGDMAPT
SCHEMBL5750943 0.70 MEN1 (0.51) NPC1RAB9AHPGDTP53SMN1; SMN2
SCHEMBL4034379 0.70 MTNR1A (0.30) MTNR1AMTNR1B
SCHEMBL4028828 0.70 CYP17A1 (0.40)
SCHEMBL8128999 0.69 KDM4E (0.39) HPGDSMN1; SMN2MTNR1AMTNR1BMAPT
SCHEMBL5752322 0.68 L3MBTL1 (0.41) RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222174-B1 IMIDAZOL-4-YLMETHANOLS USED AS INHIBITORS OF STEROID C17-20 LYASE TAKEDA PHARMACEUTICAL (JP) 2009-05-27 EP disclosed
US-6649643-B1 Antitumor, anticarcinogenic, and antimetastasis agents; benign prostatic hyperplasia, alopecia, endometriosis, uterine myoma, hirsutism, virilism, precocious puberty, mastopathy, and polycystic overay syndrome treatment TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-11-18 US disclosed
EP-1222174-A1 IMIDAZOL-4-YLMETHANOLS USED AS INHIBITORS OF STEROID C17-20 LYASE Takeda Chemical Industries, Ltd. (JP) 2002-07-17 EP disclosed
WO-2001030762-A1 IMIDAZOL-4-YLMETHANOLS USE AS INHIBITORS OF STEROID C17-20 LYASE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-03 WO disclosed