SCHEMBL4024487

SCHEMBL4024487

O=C(c1ccc2cc3c(cc2c1)CCO3)c1c[nH]cn1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCI P41743 1/20 0.35
PLA2G10 O15496 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
HDAC3 O15379 3/20 0.34
HDAC1 Q13547 3/20 0.34
HDAC2 Q92769 3/20 0.34
HDAC8 Q9BY41 3/20 0.34
HDAC6 Q9UBN7 3/20 0.34
EGLN1 Q9GZT9 1/20 0.34
MAPT P10636 2/20 0.33
MEN1 O00255 1/20 0.33
MAPK1 P28482 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
LTC4S Q16873 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
MAPK14 Q16539 1/20 0.33
TAS1R3 Q7RTX0 2/20 0.32
TAS1R1 Q7RTX1 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4030413 0.81 NPC1 (0.32) NPC1RAB9AHDAC3HDAC1HDAC2
SCHEMBL4034041 0.76 NPC1 (0.36) NPC1RAB9AMAPTSMN1; SMN2CTNNB1
SCHEMBL5750943 0.76 MEN1 (0.51) NPC1RAB9AMAPTMEN1MAPK1
SCHEMBL4030502 0.73 HDAC3 (0.34) PRKCIHDAC3HDAC1HDAC2HDAC8
SCHEMBL5678124 0.73 CYP1A2 (0.44) MAPT
SCHEMBL5678286 0.71 KDM4E (0.53) NPC1MAPTMEN1KMT2A
SCHEMBL4033986 0.71 PRKAB2 (0.41) PLA2G10NPC1RAB9AHDAC3HDAC1
SCHEMBL4028339 0.68 RAB9A (0.49) NPC1RAB9AMAPTMEN1MAPK1
SCHEMBL7266762 0.68 CYP17A1 (0.42)
SCHEMBL4024232 0.67 CTNNB1 (0.33) RAB9AMAPTMEN1KMT2ACTNNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222174-B1 IMIDAZOL-4-YLMETHANOLS USED AS INHIBITORS OF STEROID C17-20 LYASE TAKEDA PHARMACEUTICAL (JP) 2009-05-27 EP disclosed
US-6649643-B1 Antitumor, anticarcinogenic, and antimetastasis agents; benign prostatic hyperplasia, alopecia, endometriosis, uterine myoma, hirsutism, virilism, precocious puberty, mastopathy, and polycystic overay syndrome treatment TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-11-18 US disclosed
EP-1222174-A1 IMIDAZOL-4-YLMETHANOLS USED AS INHIBITORS OF STEROID C17-20 LYASE Takeda Chemical Industries, Ltd. (JP) 2002-07-17 EP disclosed
WO-2001030762-A1 IMIDAZOL-4-YLMETHANOLS USE AS INHIBITORS OF STEROID C17-20 LYASE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-03 WO disclosed