SCHEMBL4034241

SCHEMBL4034241

CCCOc1ccc(C#CCN(C)[C@H](C)[C@@H](C)O)cc1C(=O)NC(C)(O)Cc1c[nH]c2ccc(F)cc12

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 1/20 0.36
HTR1A P08908 3/20 0.35
CYP2D6 P10635 1/20 0.35
SLC6A4 P31645 2/20 0.34
SCN8A Q9UQD0 1/20 0.33
SCN10A Q9Y5Y9 1/20 0.33
ANO1 Q5XXA6 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
HTR2A P28223 4/20 0.33
HTR2C P28335 1/20 0.33
MPO P05164 2/20 0.32
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32
NOTUM Q6P988 1/20 0.32
CCKBR P32239 1/20 0.32
TACR1 P25103 1/20 0.32
SPR P35270 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4035538 0.89 ADAM17 (0.38) ADAM17HTR1ACYP2D6SLC6A4SCN8A
SCHEMBL4031721 0.86 HTR1A (0.39) ADAM17HTR1ACYP2D6SLC6A4SCN8A
SCHEMBL3937265 0.86 ADAM17 (0.36) ADAM17HTR1ASLC6A4SCN8ASCN10A
SCHEMBL13902846 0.86 ADAM17 (0.36) ADAM17HTR1ASLC6A4SCN8ASCN10A
SCHEMBL4034238 0.83 SCN8A (0.34) ADAM17HTR1ASLC6A4SCN8ASCN10A
SCHEMBL4033963 0.82 MPO (0.46) ADAM17HTR1ACYP2D6SLC6A4SCN8A
SCHEMBL4029370 0.80 HTR1A (0.42) HTR1ASLC6A4SCN8ASCN10AANO1
SCHEMBL13902841 0.77 ADAM17 (0.39) ADAM17HTR1ASLC6A4SCN8ASCN10A
SCHEMBL3943985 0.77 ADAM17 (0.39) ADAM17HTR1ASLC6A4SCN8ASCN10A
SCHEMBL3943920 0.74 ADAM17 (0.39) ADAM17HTR1ASLC6A4SCN8ASCN10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2019102-A1 Alkylacetylene substituted Acyltryptophanols Bayer Schering Pharma AG (DE) 2009-01-28 EP disclosed