SCHEMBL4035954

SCHEMBL4035954

O=C(ON1CCNCC1)c1cccc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.46
HTR3E A5X5Y0 1/20 0.46
HTR3B O95264 1/20 0.46
CYP1A2 P05177 1/20 0.46
HTR1A P08908 1/20 0.46
CYP2D6 P10635 1/20 0.46
NCF1 P14598 1/20 0.46
TSHR P16473 1/20 0.46
NFKB1 P19838 1/20 0.46
HTR1D P28221 1/20 0.46
HTR1B P28222 1/20 0.46
HTR2A P28223 1/20 0.46
HTR7 P34969 1/20 0.46
MTOR P42345 1/20 0.46
HTR3A P46098 1/20 0.46
HTR5A P47898 1/20 0.46
HTR3D Q70Z44 1/20 0.46
HTR3C Q8WXA8 1/20 0.46
HSD17B10 Q99714 1/20 0.46
SIGMAR1 Q99720 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4451473 0.86 POLB (0.54) SIGMAR1POLBGAAKMT2ALMNA
SCHEMBL5874855 0.86 RXFP1 (0.47) HTR6HTR3EHTR3BTSHRHTR3A
SCHEMBL10714629 0.85 POLB (0.56) SIGMAR1POLBGAAKMT2ALMNA
SCHEMBL5875374 0.80 TSHR (0.47) TSHRHSD17B10SIGMAR1GAAKMT2A
SCHEMBL27892691 0.79 HTT (0.44) HTR7SIGMAR1KMT2ALMNAALDH1A1
SCHEMBL3576603 0.77 ALDH1A1 (0.62) SIGMAR1POLBKMT2ALMNAALDH1A1
SCHEMBL29004525 0.77 ADRB1 (0.46) CYP1A2HTR1ACYP2D6HTR3AKMT2A
Hydrochloric Acid SCHEMBL9035292 0.76 ALDH1A1 (0.61) SIGMAR1POLBKMT2ALMNAALDH1A1
Hydrochloric Acid SCHEMBL1193388 0.76 ALDH1A1 (0.61) SIGMAR1POLBKMT2ALMNAALDH1A1
SCHEMBL24120719 0.74 SIGMAR1 (0.56) HTR6HTR3EHTR3BTSHRHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010519-A2 SUBSTITUTED IMIDAZOLE 4-CARBOXAMIDES AS CHOLECYSTOKININ-1 RECEPTOR MODULATORS Merck & Co., Inc. (US) 2009-01-07 EP disclosed
WO-2007120655-A2 SUBSTITUTED IMIDAZOLE 4-CARBOXAMIDES AS CHOLECYSTOKININ-1 RECEPTOR MODULATORS MERCK & CO., INC. (US) 2007-10-25 WO disclosed