SCHEMBL4036013

SCHEMBL4036013

O=C(O)c1c(F)csc1Br

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.47
ANO1 Q5XXA6 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
GPR35 Q9HC97 5/20 0.32
ALAD P13716 1/20 0.32
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31
DAO P14920 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL623033 0.79 TSHR (0.52) TSHRGPR35ALADCES2CES1
SCHEMBL18701591 0.77 MEN1 (0.34) TSHRANO1MEN1KMT2ACES2
SCHEMBL28196417 0.76 TSHR (0.65) TSHRKMT2AGPR35ALADCES2
SCHEMBL17398273 0.74 TSHR (0.47) TSHRMEN1KMT2AGPR35DAO
SCHEMBL18701622 0.74 KEAP1 (0.38) ANO1MEN1KMT2AGPR35ALAD
SCHEMBL2001851 0.71 TSHR (0.44) TSHRMEN1KMT2AGPR35CES2
SCHEMBL6861221 0.66
SCHEMBL19085034 0.65 TSHR (0.42) TSHRGPR35DAO
SCHEMBL516974 0.65 DGAT1 (0.42) GPR35
SCHEMBL16414224 0.64 TSHR (0.40) TSHRMEN1KMT2AGPR35CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029572-A2 ORGANIC COMPOUNDS Novartis AG (CH) 2009-03-04 EP disclosed
WO-2007143597-A2 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2007-12-13 WO disclosed