SCHEMBL4036732

SCHEMBL4036732

COc1cc(C=O)c(-c2cc(-c3nccs3)cnc2NCc2ccccc2)c(OC)c1OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 2/20 0.41
CYP1A2 P05177 6/20 0.39
CYP2D6 P10635 6/20 0.39
CYP3A4 P08684 5/20 0.39
TSHR P16473 5/20 0.39
HSD17B10 Q99714 5/20 0.39
CLK4 Q9HAZ1 3/20 0.39
ALOX15 P16050 2/20 0.39
EGFR P00533 5/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
CYP2C19 P33261 5/20 0.37
ALDH1A1 P00352 4/20 0.37
CYP2C9 P11712 3/20 0.37
MAPK1 P28482 3/20 0.37
LMNA P02545 2/20 0.37
HIF1A Q16665 2/20 0.37
USP2 O75604 1/20 0.37
HPGD P15428 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4036344 0.80 SMPD3 (0.41) TSHREGFRPTGDR2LMNASMN1; SMN2
SCHEMBL1308980 0.79 SMPD3 (0.40) TSHREGFRALDH1A1LMNASMN1; SMN2
SCHEMBL1306317 0.77 TUBB4A (0.47) PDE5ALMNAHPGDSMN1; SMN2MAPT
SCHEMBL4034103 0.75 SMPD3 (0.40) TSHRPTGDR2LMNAMAPT
SCHEMBL4034089 0.74 SMPD3 (0.46) TSHRPTGDR2LMNASMN1; SMN2MAPT
SCHEMBL4042076 0.74 MAPT (0.39) TSHREGFRPTGDR2MAPTFGFR1
SCHEMBL4034301 0.74 GABRA1 (0.41) PTGDR2ALDH1A1MAPT
SCHEMBL4042546 0.74 MAPT (0.43) TSHREGFRPTGDR2MAPTFGFR1
SCHEMBL4040171 0.73 TUBB4A (0.41) TSHRPTGDR2ALDH1A1LMNAMAPT
SCHEMBL15225671 0.73 SMPD3 (0.40) TSHRPTGDR2LMNASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2086942-A2 NOVEL COMPOUNDS Glaxo Group Limited (GB) 2009-08-12 EP disclosed
WO-2008043788-A2 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2008-04-17 WO disclosed