SCHEMBL4036984

SCHEMBL4036984

O=C(NC1CCc2ccccc21)C1CN(C(=O)Nc2ccccc2-c2ccccc2)CCN1S(=O)(=O)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
POLB P06746 1/20 0.45
HTT P42858 1/20 0.45
GAA P10253 2/20 0.43
PKM P14618 1/20 0.43
USP2 O75604 1/20 0.40
KMT2A Q03164 1/20 0.40
MMP1 P03956 1/20 0.40
MMP9 P14780 1/20 0.40
MMP13 P45452 1/20 0.40
SMO Q99835 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4034864 0.80 ALDH1A1 (0.52) ALDH1A1POLBHTTGAAPKM
SCHEMBL6190434 0.79 GAA (0.48) ALDH1A1POLBHTTGAAPKM
SCHEMBL4032820 0.72 GAA (0.49) ALDH1A1GAAMMP1MMP9MMP13
SCHEMBL4034991 0.71 GHSR (0.48) MMP1MMP9MMP13
SCHEMBL2707026 0.69 MMP1 (0.59) ALDH1A1POLBHTTGAAUSP2
SCHEMBL5244514 0.69 ALDH1A1 (0.72) ALDH1A1POLBHTTGAAPKM
SCHEMBL4033382 0.69 POLB (0.43) ALDH1A1POLBHTTGAAPKM
SCHEMBL9517197 0.68 ALDH1A1 (0.56) ALDH1A1POLBGAAKMT2ASMO
SCHEMBL6228643 0.66 OPRM1 (0.43) ALDH1A1HTTSMO
SCHEMBL4033401 0.65 MMP1 (0.54) ALDH1A1POLBHTTGAAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1592389-B1 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES SERONO LAB (CH) 2009-04-22 EP disclosed