SCHEMBL4037009

SCHEMBL4037009

COc1ccc(S(=O)(=O)N2CCN(S(=O)(=O)c3cccc4cccnc34)C(C(=O)NCCCc3ccccc3)C2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
MAPK1 P28482 2/20 0.52
MMP1 P03956 4/20 0.51
MMP3 P08254 4/20 0.51
MMP7 P09237 4/20 0.51
MMP9 P14780 4/20 0.51
HPGD P15428 1/20 0.51
GAA P10253 2/20 0.51
HTT P42858 1/20 0.51
MMP13 P45452 3/20 0.50
KMT2A Q03164 2/20 0.50
MEN1 O00255 1/20 0.50
LMNA P02545 2/20 0.49
POLB P06746 2/20 0.49
HSP90AA1 P07900 1/20 0.49
MAPT P10636 1/20 0.49
ALOX15 P16050 1/20 0.49
HSD17B10 Q99714 1/20 0.49
FKBP1A P62942 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4037013 0.87 MMP1 (0.53) ALDH1A1MMP1MMP3MMP7MMP9
SCHEMBL4034739 0.85 GAA (0.53) ALDH1A1SMN1; SMN2MAPK1MMP1MMP3
SCHEMBL1382163 0.80 GAA (0.50) ALDH1A1SMN1; SMN2HPGDGAAHTT
SCHEMBL1381140 0.80 GAA (0.50) ALDH1A1SMN1; SMN2HPGDGAAHTT
SCHEMBL4033204 0.80 GAA (0.50) ALDH1A1SMN1; SMN2HPGDGAAHTT
SCHEMBL4033581 0.78 GAA (0.57) ALDH1A1MAPK1HPGDGAAHTT
SCHEMBL4036669 0.77 ALDH1A1 (0.49) ALDH1A1MAPK1HPGDGAA
SCHEMBL4032274 0.77 GAA (0.55) ALDH1A1SMN1; SMN2MAPK1HPGDGAA
SCHEMBL1382478 0.77 ALDH1A1 (0.53) ALDH1A1MAPK1HPGDGAAKMT2A
SCHEMBL4034935 0.77 ALDH1A1 (0.51) ALDH1A1SMN1; SMN2MAPK1MMP1MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1592389-B1 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES SERONO LAB (CH) 2009-04-22 EP claimed