SCHEMBL4037899

SCHEMBL4037899

C#Cc1cccc(NC(=O)Nc2cc(C)on2)c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.70
MEN1 O00255 4/20 0.62
KMT2A Q03164 4/20 0.62
LMNA P02545 2/20 0.62
MAPK1 P28482 1/20 0.62
RAB9A P51151 6/20 0.60
SMN1; SMN2 Q16637 4/20 0.59
NPC1 O15118 4/20 0.59
L3MBTL1 Q9Y468 2/20 0.59
CYP1A2 P05177 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
MAPT P10636 4/20 0.54
HSD17B10 Q99714 1/20 0.54
KDM4E B2RXH2 2/20 0.52
POLB P06746 1/20 0.51
GAA P10253 1/20 0.51
ALOX15 P16050 1/20 0.51
IDH1 O75874 1/20 0.51
GFER P55789 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4718073 0.84 KMT2A (0.69) MEN1KMT2ARAB9ANPC1MAPT
SCHEMBL4749975 0.82 MEN1 (0.60) ALDH1A1MEN1KMT2ALMNARAB9A
SCHEMBL3939402 0.81 ALDH1A1 (0.77) ALDH1A1MEN1KMT2ALMNAMAPK1
SCHEMBL3939400 0.81 ALDH1A1 (0.77) ALDH1A1MEN1KMT2ALMNAMAPK1
SCHEMBL5728822 0.81 RAB9A (0.77) ALDH1A1MEN1KMT2ALMNAMAPK1
SCHEMBL4718568 0.80 ALDH1A1 (0.60) ALDH1A1MEN1KMT2ALMNAMAPK1
SCHEMBL13169441 0.78 IDH1 (0.57) ALDH1A1MEN1KMT2AMAPK1RAB9A
SCHEMBL12049693 0.76 IDH1 (0.54) ALDH1A1MEN1KMT2ALMNAMAPK1
SCHEMBL1025225 0.74 MEN1 (0.56) ALDH1A1MEN1KMT2ALMNARAB9A
SCHEMBL9817301 0.74 ALDH1A1 (0.65) ALDH1A1MEN1KMT2ALMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100536-A1 INHIBITORS OF KINASE ACTIVITY WITH 1,2-DI-CYCLYL SUBSTITUTED ALKYNE STRUCTURES METHYLGENE INC. (CA) 2009-08-20 WO disclosed
WO-2009100536-A1 INHIBITORS OF KINASE ACTIVITY WITH 1,2-DI-CYCLYL SUBSTITUTED ALKYNE STRUCTURES METHYLGENE INC. (CA) 2009-08-20 WO disclosed