SCHEMBL4038402

SCHEMBL4038402

COc1ccc(NC(=O)OC(C)(C)C)c(OC)c1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
GAA P10253 1/20 0.46
KDM4E B2RXH2 2/20 0.44
TSHR P16473 2/20 0.42
NR1I2 O75469 1/20 0.40
PIK3CD O00329 1/20 0.39
ABL1 P00519 1/20 0.39
EGFR P00533 1/20 0.39
KDR P35968 1/20 0.39
PIK3CA P42336 1/20 0.39
PIK3CG P48736 1/20 0.39
BACE1 P56817 1/20 0.39
PRKDC P78527 1/20 0.39
PI4KB Q9UBF8 1/20 0.39
DPP4 P27487 1/20 0.39
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
MAPK1 P28482 1/20 0.38
KMT2A Q03164 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1097144 0.86 BRD4 (0.49) ALDH1A1GAAKDM4EKMT2ANPSR1
SCHEMBL10810203 0.85 ALDH1A1 (0.42) ALDH1A1GAAKDM4ETSHRNR1I2
SCHEMBL5305447 0.85 ALDH1A1 (0.42) ALDH1A1GAAKDM4ETSHRNR1I2
SCHEMBL19932183 0.79 TAS1R3 (0.42) ALDH1A1GAAKDM4EMEN1MAPK1
SCHEMBL27625374 0.78 TDP1 (0.47) ALDH1A1GAAKDM4ETSHRMEN1
SCHEMBL15457550 0.78 EPHX1 (0.57) ALDH1A1GAAPIK3CDABL1EGFR
SCHEMBL729221 0.78 KMT2A (0.59) ALDH1A1GAAKDM4EMEN1MAPK1
SCHEMBL29991357 0.78 KMT2A (0.59) ALDH1A1GAAKDM4EMEN1MAPK1
SCHEMBL2589170 0.77 ALDH1A1 (0.63) ALDH1A1GAAKDM4ETSHRMEN1
SCHEMBL30087033 0.77 HSP90AA1 (0.45) ALDH1A1GAAMEN1KMT2APKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562589-B1 DIAMINOTRIAZOLES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2009-01-07 EP disclosed