SCHEMBL4040753

SCHEMBL4040753

Nc1nc(Nc2cccc3c2OC(F)(F)O3)nn1-c1cc(Cl)ncn1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 7/20 0.43
IRAK4 Q9NWZ3 6/20 0.43
AURKA O14965 2/20 0.43
KIT P10721 5/20 0.39
BACE1 P56817 4/20 0.37
ADORA2A P29274 3/20 0.35
JAK2 O60674 2/20 0.35
SRC P12931 1/20 0.35
CDK2 P24941 1/20 0.35
ATR Q13535 1/20 0.35
JAK3 P52333 1/20 0.34
PTK2 Q05397 1/20 0.34
DOT1L Q8TEK3 1/20 0.34
AXL P30530 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4044453 0.82 FLT3 (0.59) FLT3IRAK4AURKAKITADORA2A
SCHEMBL4039634 0.74 FLT3 (0.45) FLT3IRAK4AURKAKITJAK2
SCHEMBL4040322 0.74 FLT3 (0.67) FLT3IRAK4AURKAKITJAK2
SCHEMBL4046935 0.73 FLT3 (0.45) FLT3IRAK4AURKAKITBACE1
SCHEMBL2086579 0.73 FLT3 (0.48) FLT3IRAK4AURKAKITBACE1
SCHEMBL6224723 0.69 ULK1 (0.44) FLT3IRAK4AURKAKITBACE1
SCHEMBL4043796 0.68 FLT3 (0.61) FLT3IRAK4AURKAKITJAK2
SCHEMBL13963975 0.68 AXL (0.44) FLT3IRAK4AURKAKITBACE1
SCHEMBL12782391 0.67 FLT3 (0.44) FLT3IRAK4AURKAKITBACE1
SCHEMBL20260472 0.67 BACE1 (0.38) BACE1ADORA2AJAK2SRCCDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562589-B1 DIAMINOTRIAZOLES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2009-01-07 EP disclosed