SCHEMBL4042434

SCHEMBL4042434

Cc1cccc(Cl)c1-c1cc(NCCO)nc2c1nc(N)c1cncn12

nearest known ligand 0.41

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
LCK P06239 19/20 0.41
FGFR1 P11362 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4042263 0.89 LCK (0.47) LCKFGFR1
SCHEMBL4036111 0.87 LCK (0.42) LCKFGFR1
SCHEMBL4044486 0.85 LCK (0.38) LCK
SCHEMBL4041190 0.85 LCK (0.51) LCKFGFR1
SCHEMBL4037168 0.84 MEN1 (0.44) LCKFGFR1
SCHEMBL4043849 0.82 LCK (0.43) LCKFGFR1
SCHEMBL4042428 0.82 LCK (0.44) LCKFGFR1
SCHEMBL4036365 0.81 FGFR1 (0.40) LCKFGFR1
SCHEMBL4038945 0.79 LCK (0.50) LCK
SCHEMBL4040159 0.78 LCK (0.38) LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1066286-B1 HETEROCYCLO-SUBSTITUTED IMIDAZOPYRAZINE PROTEIN TYROSINE KINASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2009-04-29 EP claimed
EP-1066286-B1 HETEROCYCLO-SUBSTITUTED IMIDAZOPYRAZINE PROTEIN TYROSINE KINASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2009-04-29 EP disclosed