SCHEMBL4043183

SCHEMBL4043183

CC(C)CC(NC(=O)Oc1ccc2ccccc2c1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)C(=O)c1cccnc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 8/20 0.43
MMP1 P03956 1/20 0.39
MMP3 P08254 1/20 0.39
MMP9 P14780 1/20 0.39
ELANE P08246 1/20 0.36
CYP3A4 P08684 3/20 0.36
CYP2C9 P11712 3/20 0.36
CYP2C19 P33261 3/20 0.36
MC4R P32245 1/20 0.35
MC3R P41968 1/20 0.35
MC1R Q01726 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
ALDH1A1 P00352 2/20 0.33
CYP1A2 P05177 2/20 0.33
CTSL P07711 2/20 0.33
CTSB P07858 2/20 0.33
CTSS P25774 2/20 0.33
LMNA P02545 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4039893 0.93 CTSK (0.41) CTSKMMP1MMP3MMP9ELANE
SCHEMBL4051965 0.93 MC4R (0.38) CTSKMMP1MMP3MMP9ELANE
SCHEMBL4045571 0.92 CTSK (0.46) CTSKMMP1MMP3MMP9ELANE
SCHEMBL4040677 0.90 CTSK (0.41) CTSKMMP1MMP3MMP9SMN1; SMN2
SCHEMBL4039972 0.89 CTSK (0.40) CTSKMMP1MMP3MMP9ELANE
SCHEMBL4042370 0.89 CTSK (0.42) CTSKMMP1MMP3MMP9ELANE
SCHEMBL4041363 0.89 CTSK (0.42) CTSKMMP1MMP3MMP9ELANE
SCHEMBL4045633 0.88 CTSK (0.41) CTSKMMP1MMP3MMP9ALDH1A1
SCHEMBL4045591 0.88 CTSK (0.41) CTSKMMP1MMP3MMP9ELANE
SCHEMBL4047118 0.88 CTSK (0.41) CTSKMMP1MMP3MMP9ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed