SCHEMBL4045571

SCHEMBL4045571

CC(C)CC(NC(=O)Oc1ccc(-c2ccccc2)cc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)C(=O)c1cccnc1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSK P43235 13/20 0.46
ELANE P08246 1/20 0.39
MMP1 P03956 1/20 0.37
MMP3 P08254 1/20 0.37
MMP9 P14780 1/20 0.37
CTSL P07711 6/20 0.35
CTSS P25774 5/20 0.35
CTSB P07858 2/20 0.35
HRH3 Q9Y5N1 1/20 0.34
PREP P48147 1/20 0.34
FAP Q12884 1/20 0.34
CHRNA7 P36544 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043596 0.92 ELANE (0.38) CTSKELANEMMP1MMP3MMP9
SCHEMBL4043183 0.92 CTSK (0.43) CTSKELANEMMP1MMP3MMP9
SCHEMBL4042585 0.90 USP30 (0.39) CTSKELANE
SCHEMBL4051777 0.89 CTSK (0.44) CTSKELANEMMP1MMP3MMP9
SCHEMBL4045331 0.89 CTSK (0.43) CTSKELANEMMP1MMP3MMP9
SCHEMBL4042529 0.89 BCL2 (0.38) CTSKELANE
SCHEMBL4045591 0.89 CTSK (0.41) CTSKELANEMMP1MMP3MMP9
SCHEMBL4047118 0.89 CTSK (0.41) CTSKELANEMMP1MMP3MMP9
SCHEMBL4043465 0.89 MC4R (0.41) CTSKELANE
SCHEMBL4041055 0.88 CTSK (0.49) CTSKCTSLCTSSCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed