SCHEMBL4051965

SCHEMBL4051965

CCCC(NC(=O)Oc1ccc2ccccc2c1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)C(=O)c1cccnc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MC4R P32245 1/20 0.38
MC3R P41968 1/20 0.38
MC1R Q01726 1/20 0.38
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
CTSK P43235 6/20 0.35
CCR1 P32246 1/20 0.35
ROCK2 O75116 1/20 0.34
MMP1 P03956 1/20 0.34
MMP3 P08254 1/20 0.34
MMP9 P14780 1/20 0.34
ELANE P08246 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KLK7 P49862 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
TACR1 P25103 1/20 0.32
GPR132 Q9UNW8 3/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4044339 0.94 ALDH1A1 (0.37) MC4RMC3RMC1RCTSKMMP1
SCHEMBL4043183 0.93 CTSK (0.43) MC4RMC3RMC1RCYP3A4CYP2C9
SCHEMBL4043596 0.92 ELANE (0.38) MC4RMC3RMC1RCYP3A4CYP2C9
SCHEMBL4044730 0.90 LMNA (0.39) CTSKCCR1ROCK2MMP1MMP3
SCHEMBL4043124 0.90 POLB (0.34) CTSKELANESMN1; SMN2RXFP1KDM4E
SCHEMBL4045687 0.89 MC4R (0.34) MC4RMC3RMC1RCTSKCCR1
SCHEMBL4042570 0.89 CTSK (0.34) MC4RMC3RMC1RCTSKMMP1
SCHEMBL4046940 0.88 KDM4E (0.35) MC4RMC3RMC1RCTSKMMP1
SCHEMBL4045553 0.88 CTSK (0.34) MC4RMC3RMC1RCTSKELANE
SCHEMBL4047844 0.88 SMYD3 (0.35) MC4RMC3RMC1RCTSKTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed